SCHEMBL7965539

SCHEMBL7965539

O=[N+]([O-])c1ccc2ccc(C3CCNCC3)nc2c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
CYP3A4 P08684 2/20 0.46
HTR3E A5X5Y0 1/20 0.46
HTR3B O95264 1/20 0.46
CYP1A2 P05177 1/20 0.46
SLC6A4 P31645 1/20 0.46
CYP2C19 P33261 1/20 0.46
THPO P40225 1/20 0.46
HTR3A P46098 1/20 0.46
HTR3D Q70Z44 1/20 0.46
HTR3C Q8WXA8 1/20 0.46
RAB9A P51151 1/20 0.43
CHRNB4 P30926 2/20 0.40
CHRNA3 P32297 2/20 0.40
MAPT P10636 2/20 0.40
GABRA1 P14867 1/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
LMNA P02545 2/20 0.40
PMP22 Q01453 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31703587 0.80 RAB9A (0.61) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL31458446 0.80 ALDH1A1 (0.50) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL7966522 0.78 CYP3A4 (0.44) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL7970193 0.77 ALDH1A1 (0.48) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL7955026 0.75 MEN1 (0.42) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL19411398 0.75 BACE1 (0.43) CYP1A2SLC6A4CYP2C19RAB9A
SCHEMBL7968273 0.75 KMT2A (0.57) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL7970187 0.74 ALDH1A1 (0.56) ALDH1A1CYP3A4CYP1A2RAB9AMAPT
SCHEMBL29733200 0.72 MEN1 (0.57) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2
SCHEMBL21000902 0.72 MEN1 (0.57) ALDH1A1CYP3A4HTR3EHTR3BCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed