SCHEMBL7966522

SCHEMBL7966522

O=[N+]([O-])c1ccc2cc(C3CCNCC3)ncc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.44
ALDH1A1 P00352 2/20 0.44
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
CYP1A2 P05177 1/20 0.44
SLC6A4 P31645 1/20 0.44
CYP2C19 P33261 1/20 0.44
THPO P40225 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
MAPT P10636 2/20 0.40
NOS1 P29475 2/20 0.40
LMNA P02545 2/20 0.40
ALOX15 P16050 1/20 0.40
POLB P06746 1/20 0.40
MAOB P27338 1/20 0.40
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7965539 0.78 ALDH1A1 (0.46) CYP3A4ALDH1A1HTR3EHTR3BCYP1A2
SCHEMBL7955491 0.76 L3MBTL1 (0.40) SLC6A4HTR3ANOS1GABRA1RAB9A
SCHEMBL5241881 0.75 BCHE (0.45) CYP1A2SLC6A4HTR3AGABRA1
Hydrochloric Acid SCHEMBL3880186 0.74 BCHE (0.44) CYP1A2SLC6A4HTR3AGABRA1
SCHEMBL10834084 0.71 HRH4 (0.46) CYP1A2SLC6A4HTR3AGABRA1
SCHEMBL31703587 0.70 RAB9A (0.61) CYP3A4ALDH1A1HTR3EHTR3BCYP1A2
SCHEMBL7970187 0.69 ALDH1A1 (0.56) CYP3A4ALDH1A1CYP1A2MAPTLMNA
SCHEMBL7970193 0.69 ALDH1A1 (0.48) CYP3A4ALDH1A1HTR3EHTR3BCYP1A2
SCHEMBL7955486 0.69 BCHE (0.57) CYP3A4ALDH1A1HTR3EHTR3BCYP1A2
SCHEMBL17374976 0.69 MAPT (0.46) CYP3A4ALDH1A1CYP1A2MAPTNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
WO-1999065487-A1 INHIBITORS OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed