SCHEMBL7965613

SCHEMBL7965613

OCc1cc(-c2ccccn2)nc2ccccc12

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.55
CYP3A4 P08684 2/20 0.55
METAP1 P53582 4/20 0.54
CBFB Q13951 1/20 0.52
KDM4E B2RXH2 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
DHODH Q02127 1/20 0.51
NPSR1 Q6W5P4 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
MAPK1 P28482 2/20 0.49
ADORA3 P0DMS8 1/20 0.49
ALOX15 P16050 1/20 0.48
TSHR P16473 1/20 0.48
HSD17B10 Q99714 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
PKM P14618 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8338056 0.86 METAP1 (0.48) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL13243235 0.85 CYP3A4 (0.53) CYP2C9CYP3A4METAP1KDM4ERXFP1
SCHEMBL8335864 0.85 CBFB (0.46) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL8336808 0.85 NPSR1 (0.46) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL8333690 0.85 CBFB (0.46) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL8333603 0.85 CCR1 (0.51) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL8334580 0.85 NPC1 (0.47) CYP2C9CYP3A4METAP1CBFBKDM4E
SCHEMBL8336614 0.85 KDM4E (0.54) CYP2C9CYP3A4METAP1KDM4EDHODH
SCHEMBL7952415 0.84 CYP2C9 (0.56) CYP2C9CYP3A4METAP1KDM4EDHODH
SCHEMBL7962384 0.83 CYP3A4 (0.57) CYP2C9CYP3A4METAP1CBFBDHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed
US-5874587-A FLUORESCENCE THE ROCKEFELLER UNIVERSITY (US) 1999-02-23 US disclosed