SCHEMBL7962384

SCHEMBL7962384

OCc1cc(-c2cnccn2)nc2ccccc12

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.57
METAP2 P50579 1/20 0.47
PIM1 P11309 1/20 0.42
NPSR1 Q6W5P4 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MEN1 O00255 1/20 0.40
CACNA1B Q00975 1/20 0.40
APBA1 Q02410 1/20 0.40
KMT2A Q03164 1/20 0.40
CBFB Q13951 1/20 0.40
DHODH Q02127 3/20 0.39
CYP2C9 P11712 3/20 0.39
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
METAP1 P53582 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7965613 0.83 CYP2C9 (0.55) CYP3A4NPSR1TDP1CBFBDHODH
SCHEMBL4007503 0.79 CYP3A4 (0.73) CYP3A4MEN1KMT2ADHODH
SCHEMBL26649767 0.76 DHODH (0.60) CYP3A4NPSR1MEN1KMT2ADHODH
SCHEMBL7967523 0.76 CYP3A4 (0.60) CYP3A4NPSR1TDP1MEN1CACNA1B
SCHEMBL1259674 0.75 ACHE (0.59) DHODHCYP2C9
SCHEMBL321962 0.74 METAP2 (0.54) CYP3A4METAP2PIM1NPSR1TDP1
SCHEMBL29660606 0.74 METAP2 (0.54) CYP3A4METAP2PIM1NPSR1TDP1
SCHEMBL14734857 0.74 METAP2 (0.50) CYP3A4METAP2PIM1KMT2ADHODH
SCHEMBL6078617 0.72 ADRA1A (0.43) METAP2
SCHEMBL8272308 0.72 CYP3A4 (0.47) CYP3A4METAP2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed