SCHEMBL7952415

SCHEMBL7952415

O=C(O)Cc1cc(-c2ccccn2)nc2ccccc12

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.56
CYP3A4 P08684 2/20 0.56
ADORA3 P0DMS8 1/20 0.54
DHODH Q02127 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
TDP1 Q9NUW8 1/20 0.53
MAPK1 P28482 2/20 0.51
ALDH1A1 P00352 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
PKM P14618 1/20 0.50
KDM4E B2RXH2 1/20 0.50
METAP1 P53582 1/20 0.50
ALOX15 P16050 1/20 0.50
TSHR P16473 1/20 0.50
HSD17B10 Q99714 1/20 0.50
LMNA P02545 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.49
MAPT P10636 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8334151 0.88 ADORA3 (0.46) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL8335356 0.87 KDM4E (0.52) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL8334494 0.87 KMT2A (0.48) CYP2C9CYP3A4ADORA3NPSR1TDP1
SCHEMBL8335971 0.87 ADORA3 (0.45) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL8335315 0.87 ADORA3 (0.45) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL8335283 0.87 NPSR1 (0.51) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL7965613 0.84 CYP2C9 (0.55) CYP2C9CYP3A4ADORA3DHODHNPSR1
SCHEMBL13243235 0.83 CYP3A4 (0.53) CYP2C9CYP3A4DHODHNPSR1TDP1
SCHEMBL8334301 0.83 METAP1 (0.49) ADORA3NPSR1KDM4EMETAP1LMNA
SCHEMBL10506477 0.81 KDM4E (0.61) CYP2C9CYP3A4DHODHTDP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed
US-5874587-A FLUORESCENCE THE ROCKEFELLER UNIVERSITY (US) 1999-02-23 US disclosed