SCHEMBL7965987

SCHEMBL7965987

FC(F)(F)c1cccc2nc(C3CCNCC3)oc12

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.49
CYP1A2 P05177 3/20 0.45
CYP2C19 P33261 2/20 0.45
SLC6A2 P23975 3/20 0.42
SLC6A4 P31645 3/20 0.42
HTR1A P08908 1/20 0.42
SLC6A3 Q01959 1/20 0.42
MPO P05164 1/20 0.40
CASP6 P55212 1/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
HRH4 Q9H3N8 1/20 0.37
C1R P00736 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23411785 0.82 MPO (0.46) SLC6A2SLC6A4HTR1ASLC6A3MPO
SCHEMBL20135544 0.79 HTR2C (0.46) HTR2CCYP1A2SLC6A2SLC6A4HTR1A
SCHEMBL204714 0.74 PARP1 (0.51) KDM4EALDH1A1
SCHEMBL2961557 0.73 HTR2C (0.49) HTR2CCYP1A2CYP2C19SLC6A2SLC6A4
SCHEMBL7966615 0.73 LMNA (0.46) HTR2CSLC6A2SLC6A4HTR1ASLC6A3
SCHEMBL373400 0.72 MPO (0.54) MPOALDH1A1MEN1KMT2APOLB
SCHEMBL7956610 0.71 HTR2C (0.50) HTR2CCYP1A2CYP2C19SLC6A2SLC6A4
SCHEMBL2709039 0.70 MPO (0.59) HTR2CMPOCASP6ALDH1A1MEN1
SCHEMBL7969690 0.70 MEN1 (0.56) HTR2CCYP1A2CYP2C19SLC6A2SLC6A4
SCHEMBL22382316 0.68 C1R (0.41) CYP1A2CYP2C19KDM4EALDH1A1C1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303627-B1 FOR THERAPY OF PHYSIOLOGICAL AND PSYCHOLOGICAL DISORDERS ELI LILLY AND COMPANY 2001-10-16 US disclosed
WO-1999065487-A1 INHIBITORS OF SEROTONIN REUPTAKE ELI LILLY AND COMPANY (US) 1999-12-23 WO disclosed
EP-0965587-A1 Tetrahydropyridinyl- and piperidinyl Inhibitors of serotonin reuptake ELI LILLY AND COMPANY (US) 1999-12-22 EP disclosed