SCHEMBL7966046

SCHEMBL7966046

CCOC(=O)c1cn(C2CCN(C(=O)OCc3ccccc3)CC2)c2ncccc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.47
MAPK1 P28482 1/20 0.47
GRIN2B Q13224 7/20 0.46
ELANE P08246 1/20 0.46
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
CYP2C19 P33261 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
NOS2 P35228 1/20 0.43
CCR8 P51685 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7963486 0.90 GRIN2B (0.50) GRIN2BSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL7962923 0.87 ELANE (0.48) TSHRMAPK1ELANESMN1; SMN2L3MBTL1
SCHEMBL7953666 0.85 ELANE (0.58) TSHRMAPK1ELANE
SCHEMBL7954726 0.85 GRIN2B (0.46) GRIN2BSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL7954870 0.85 GRIN2B (0.46) GRIN2BSMN1; SMN2NPC1RAB9ACYP2C19
SCHEMBL7960116 0.85 TSHR (0.45) TSHRMAPK1ELANEL3MBTL1
SCHEMBL7966506 0.85 TSHR (0.45) TSHRMAPK1ELANEL3MBTL1
SCHEMBL7966469 0.83 ELANE (0.56) ELANE
SCHEMBL7954868 0.83 ELANE (0.56) ELANE
SCHEMBL7946372 0.82 ELANE (0.55) MAPK1ELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331548-B1 PREVENTION OR TREATMENT OF CYTOKINE RELATED DISEASES SUNTORY LIMITED (JP) 2001-12-18 US disclosed
EP-0978516-A1 1-CYCLOALKYL-1,8-NAPHTHYRIDIN-4-ONE DERIVATIVES WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SUNTORY LIMITED (JP) 2000-02-09 EP disclosed