SCHEMBL7960116

SCHEMBL7960116

CCOC(=O)c1cn([C@H]2CC[C@H](NC(=O)OCc3ccccc3)CC2)c2ncccc2c1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.45
MAPK1 P28482 1/20 0.45
ELANE P08246 1/20 0.45
ALDH1A1 P00352 2/20 0.45
GAA P10253 1/20 0.45
ADORA2A P29274 1/20 0.43
ADORA1 P30542 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
PPIA P62937 1/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
JAK2 O60674 1/20 0.40
JAK1 P23458 1/20 0.40
TYK2 P29597 1/20 0.40
ROCK2 O75116 2/20 0.40
MAPK8 P45983 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7966506 1.00 TSHR (0.45) TSHRMAPK1ELANEALDH1A1GAA
SCHEMBL7963864 0.91 ALDH1A1 (0.48) TSHRALDH1A1GAAADORA2AADORA1
SCHEMBL7954789 0.91 ALDH1A1 (0.48) TSHRALDH1A1GAAADORA2AADORA1
SCHEMBL7954575 0.86 ELANE (0.46) ELANEALDH1A1PDE4APDE4BPDE4C
SCHEMBL7953666 0.86 ELANE (0.58) TSHRMAPK1ELANE
SCHEMBL7966046 0.85 TSHR (0.47) TSHRMAPK1ELANEL3MBTL1
SCHEMBL7961978 0.82 PDE4A (0.53) TSHRALDH1A1GAAPDE4APDE4B
SCHEMBL7961980 0.82 PDE4A (0.53) TSHRALDH1A1GAAPDE4APDE4B
SCHEMBL7960265 0.82 ELANE (0.54) ELANEMAPK8
SCHEMBL7966421 0.82 ELANE (0.54) ELANEMAPK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6331548-B1 PREVENTION OR TREATMENT OF CYTOKINE RELATED DISEASES SUNTORY LIMITED (JP) 2001-12-18 US disclosed
EP-0978516-A1 1-CYCLOALKYL-1,8-NAPHTHYRIDIN-4-ONE DERIVATIVES WITH PHOSPHODIESTERASE IV INHIBITORY ACTIVITY SUNTORY LIMITED (JP) 2000-02-09 EP disclosed