SCHEMBL7967523

SCHEMBL7967523

O=C(OCCO)c1cc(-c2cnccn2)nc2ccccc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 5/20 0.60
KDM4E B2RXH2 6/20 0.52
MEN1 O00255 4/20 0.52
KMT2A Q03164 4/20 0.52
ALDH1A1 P00352 2/20 0.52
CACNA1B Q00975 1/20 0.47
APBA1 Q02410 1/20 0.47
MAPT P10636 6/20 0.47
HPGD P15428 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TP53 P04637 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
RAB9A P51151 1/20 0.44
TDP1 Q9NUW8 2/20 0.44
POLB P06746 1/20 0.44
RECQL P46063 1/20 0.44
PLA2G2A P14555 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
DHODH Q02127 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8429927 0.87 CYP2C9 (0.58) CYP3A4KDM4EALDH1A1MAPTSMN1; SMN2
SCHEMBL28676204 0.82 KDM4E (0.62) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL4007503 0.81 CYP3A4 (0.73) CYP3A4KDM4EMEN1KMT2ASMN1; SMN2
SCHEMBL7962384 0.76 CYP3A4 (0.57) CYP3A4MEN1KMT2ACACNA1BAPBA1
SCHEMBL31310821 0.75 ALDH1A1 (0.61) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL14990402 0.75 ALDH1A1 (0.61) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL31310820 0.74 PLA2G2A (0.65) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL5400497 0.74 PLA2G2A (0.65) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL2918797 0.73 KDM4E (0.67) CYP3A4KDM4EMEN1KMT2AALDH1A1
SCHEMBL4393431 0.70 CYP3A4 (0.62) CYP3A4KDM4EMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6187928-B1 TREATING FUNGAL DISEASES THE ROCKEFELLER UNIVERSITY 2001-02-13 US disclosed
US-6087510-A Method of use of imidazolium cations THE ROCKEFELLER UNIVERSITY (US) 2000-07-11 US disclosed