SCHEMBL7968435

SCHEMBL7968435

COc1ccc(-c2nc3c(OC)cc(C)nc3[nH]2)c(OC)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.50
KDM4E B2RXH2 4/20 0.46
CYP1A2 P05177 2/20 0.46
CYP3A4 P08684 2/20 0.46
GAA P10253 3/20 0.44
HSD17B10 Q99714 2/20 0.44
MGAM O43451 2/20 0.44
SI P14410 2/20 0.44
MGAM2 Q2M2H8 2/20 0.44
TSHR P16473 1/20 0.44
HTT P42858 3/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP1A1 P04798 3/20 0.42
CYP1B1 Q16678 3/20 0.42
CRHR1 P34998 2/20 0.41
CYP2E1 P05181 1/20 0.41
CYP2C8 P10632 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2A6 P11509 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2947301 0.79 PDE2A (0.48) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL7968594 0.76 TNKS (0.50) KDM4EGAAHSD17B10MGAMSI
SCHEMBL10685704 0.75 PDE2A (0.50) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL10742148 0.74 PDE2A (0.68) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL10848799 0.74 PDE2A (0.64) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL6040494 0.72 PDE2A (0.65) PDE2AKDM4ECYP1A2CYP3A4HSD17B10
SCHEMBL7280668 0.71 PDE2A (0.57) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL10690574 0.71 PDE2A (0.51) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL11237399 0.71 PDE2A (0.51) PDE2AKDM4ECYP1A2CYP3A4GAA
SCHEMBL10847442 0.71 PDE2A (0.64) PDE2AKDM4ECYP1A2CYP3A4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003744-A1 4-AMINOPYRROLE(3,2-d) PYRIMIDINES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS Pfizer Products Inc. (US) 2000-05-31 EP claimed
WO-1999007703-A1 4-AMINOPYRROLE(3,2-d) PYRIMIDINES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 1999-02-18 WO claimed
US-6187778-B1 EATING AND CARDIOVASCULAR DISORDERS PFIZER INC. 2001-02-13 US disclosed
EP-1003744-A1 4-AMINOPYRROLE(3,2-d) PYRIMIDINES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS Pfizer Products Inc. (US) 2000-05-31 EP disclosed
WO-1999007703-A1 4-AMINOPYRROLE(3,2-d) PYRIMIDINES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. (US) 1999-02-18 WO disclosed