SCHEMBL7969464

SCHEMBL7969464

CC(=O)SCCc1nnc2ccccn12

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.53
ALDH1A1 P00352 3/20 0.53
RAB9A P51151 6/20 0.51
NPC1 O15118 5/20 0.51
SMN1; SMN2 Q16637 5/20 0.47
HPGD P15428 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 2/20 0.40
CYP2C9 P11712 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7983167 0.76 GGPS1 (0.48) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7979860 0.76 PDE10A (0.42) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7969877 0.75 ALDH1A1 (0.49) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL24273206 0.75 KDM4E (0.67) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7983003 0.75 KDM4E (0.67) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL24862850 0.75 KDM4E (0.67) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7983166 0.74 PTGS1 (0.49) KDM4EALDH1A1SMN1; SMN2TDP1LMNA
SCHEMBL5354841 0.74 KDM4E (0.56) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL7980785 0.72 KDM4E (0.62) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2
SCHEMBL5373208 0.71 KDM4E (0.71) KDM4EALDH1A1RAB9ANPC1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed