SCHEMBL7983166

SCHEMBL7983166

CC(=O)SCCc1nc2ccccn2c1N

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.49
PTGS2 P35354 1/20 0.49
KMT2A Q03164 2/20 0.43
ALDH1A1 P00352 5/20 0.42
KDM4E B2RXH2 4/20 0.42
GAA P10253 2/20 0.42
DAPK3 O43293 1/20 0.42
JAK2 O60674 1/20 0.42
PRKD3 O94806 1/20 0.42
MAP4K4 O95819 1/20 0.42
ABL1 P00519 1/20 0.42
CSF1R P07333 1/20 0.42
RET P07949 1/20 0.42
MET P08581 1/20 0.42
PDGFRA P16234 1/20 0.42
PRKACA P17612 1/20 0.42
LTK P29376 1/20 0.42
GRK5 P34947 1/20 0.42
KDR P35968 1/20 0.42
MAPK8 P45983 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969877 0.85 ALDH1A1 (0.49) KMT2AALDH1A1KDM4EGAATDP1
SCHEMBL7986214 0.77 PTGS1 (0.51) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL7969464 0.74 KDM4E (0.53) KMT2AALDH1A1KDM4ETDP1SMN1; SMN2
SCHEMBL23890512 0.74 PTGS1 (0.50) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL7983167 0.73 GGPS1 (0.48) KMT2AALDH1A1KDM4EGAASMN1; SMN2
SCHEMBL18412790 0.71 PTGS1 (0.73) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL7979455 0.71 MAPK1 (0.53) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL7980201 0.71 RAB9A (0.38) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL7969549 0.70 KDM4E (0.51) PTGS1PTGS2KMT2AALDH1A1KDM4E
SCHEMBL14078787 0.68 ALDH1A1 (0.44) PTGS1PTGS2KMT2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed