SCHEMBL7979860

SCHEMBL7979860

CC(=O)SCCc1ncc2ccccn12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.42
ALDH1A1 P00352 12/20 0.42
KDM4E B2RXH2 11/20 0.42
MAPT P10636 6/20 0.42
RAB9A P51151 6/20 0.42
HPGD P15428 6/20 0.39
CHEK1 O14757 1/20 0.39
LIMK1 P53667 1/20 0.39
MAPK14 Q16539 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
NPC1 O15118 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
HSD17B10 Q99714 3/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
SSTR4 P31391 1/20 0.36
GLA P06280 1/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7981104 0.81 SSTR4 (0.35) SSTR4POLB
SCHEMBL15491630 0.78 ALDH1A1 (0.44) PDE10AALDH1A1KDM4EMAPTRAB9A
SCHEMBL27940752 0.78 PDE10A (0.42) PDE10AALDH1A1KDM4EMAPTRAB9A
SCHEMBL7983167 0.78 GGPS1 (0.48) ALDH1A1KDM4EMAPTRAB9AHPGD
SCHEMBL7969464 0.76 KDM4E (0.53) ALDH1A1KDM4ERAB9AHPGDTDP1
SCHEMBL7983487 0.76 KDM4E (0.47) PDE10AALDH1A1KDM4EMAPTRAB9A
SCHEMBL3798563 0.76 KDM4E (0.47) PDE10AALDH1A1KDM4EMAPTRAB9A
Hydrochloric Acid SCHEMBL3795323 0.74 KDM4E (0.46) PDE10AALDH1A1KDM4EMAPTRAB9A
SCHEMBL12480176 0.73 ALDH1A1 (0.49) PDE10AALDH1A1KDM4EMAPTRAB9A
SCHEMBL7980854 0.72 KDM4E (0.38) ALDH1A1KDM4EHPGDCHEK1LIMK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed