SCHEMBL7969520

SCHEMBL7969520

Cc1cc(C(C)(C)C)ccc1CCl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PON1 P27169 1/20 0.47
HTR1D P28221 2/20 0.46
ADRA2A P08913 1/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
ADRA1D P25100 1/20 0.46
HTR1B P28222 1/20 0.46
ADRA1A P35348 1/20 0.46
ADRA1B P35368 1/20 0.46
CYP2C19 P33261 2/20 0.46
CYP1A2 P05177 1/20 0.46
TSHR P16473 1/20 0.41
EPHX2 P34913 1/20 0.41
ALDH1A1 P00352 3/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
RXRA P19793 1/20 0.40
RXRB P28702 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11223586 0.85 PON1 (0.46) PON1HTR1DADRA2AADRA2BADRA2C
SCHEMBL30617195 0.81 DAO (0.46) RXRARXRBPOLBMAPT
SCHEMBL5111503 0.81 DAO (0.46) RXRARXRBPOLBMAPT
SCHEMBL6644304 0.79 PON1 (0.45) PON1HTR1DADRA2AADRA2BADRA2C
SCHEMBL11344556 0.79 ALDH1A1 (0.57) PON1CYP2C19CYP1A2TSHRALDH1A1
SCHEMBL7979494 0.78 KLF10 (0.47) HTR1DADRA2AADRA2BADRA2CADRA1D
SCHEMBL12049340 0.78 HTR1D (0.46) HTR1DADRA2AADRA2BADRA2CADRA1D
SCHEMBL11280631 0.77 HTR1D (0.40) PON1HTR1DADRA2AADRA2BADRA2C
SCHEMBL26802829 0.77 HTR1D (0.45) HTR1DADRA2AADRA2BADRA2CADRA1D
SCHEMBL23402375 0.75 HTR1D (0.44) HTR1DADRA2AADRA2BADRA2CADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6288101-B1 ADMINISTERING COMPOUNDS SUCH AS 2,6-DIMETHYL-4-ISOPROPYLBENZALDEHYDE TO TREAT INDICATIONS WHERE STIMULATION OF SUBTYPES OF THE SEROTONIN RECEPTOR IS IMPLICATED, SUCH AS MIGRAINES VIRGINIA COMMONWEALTH UNIVERSITY 2001-09-11 US disclosed
US-6124338-A TREATING MIGRAINE HEADACHE VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-09-26 US disclosed
US-6048862-A Benzylamidine derivatives with serotonin receptor binding activity VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-04-11 US disclosed
US-5969137-A TREATMENT OF NERVOUS SYSTEM DISORDERS VIRGINIA COMMONWEALTH UNIVERSITY (US) 1999-10-19 US disclosed
WO-1998012183-A1 IMIDAZOLES WITH SEROTONIN RECEPTOR BINDING ACTIVITY ALLELIX BIOPHARMACEUTICALS INC. (CA) 1998-03-26 WO disclosed