SCHEMBL7969694

SCHEMBL7969694

Nc1nc2c(-c3c(F)cccc3Cl)cc(NCCc3ccncc3)cc2n2cncc12

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LCK P06239 6/20 0.38
NPC1 O15118 1/20 0.38
CCNT1 O60563 1/20 0.38
CDK9 P50750 1/20 0.36
ADORA2A P29274 1/20 0.36
ADORA1 P30542 1/20 0.36
MKNK2 Q9HBH9 7/20 0.36
MKNK1 Q9BUB5 4/20 0.36
CDK2 P24941 1/20 0.34
KCNK13 Q9HB14 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7979832 0.85 LCK (0.49) LCK
SCHEMBL7987033 0.83 LCK (0.49) LCKCCNT1CDK9
SCHEMBL7969619 0.83 LCK (0.37) LCKCCNT1CDK9
SCHEMBL7982995 0.82 LCK (0.47) LCKCCNT1CDK9
SCHEMBL7987540 0.82 LCK (0.46) LCKCCNT1CDK9
SCHEMBL7983616 0.81 LCK (0.51) LCKNPC1CCNT1ADORA2AADORA1
SCHEMBL7983677 0.80 FGFR1 (0.50) LCK
SCHEMBL7980019 0.80 LCK (0.52) LCK
SCHEMBL7970506 0.79 RAD52 (0.39) LCKNPC1
SCHEMBL7969601 0.78 FGFR1 (0.44) LCKCDK9ADORA2AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US claimed
WO-1999009845-A1 IMIDAZOQUINOXALINE PROTEIN TYROSINE KINASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 1999-03-04 WO claimed
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed