SCHEMBL7969955

SCHEMBL7969955

O=c1[nH]c2ccc([N+](=O)[O-])cc2n2cncc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 1/20 0.51
GRIA2 P42262 1/20 0.51
GRIA3 P42263 1/20 0.51
GRIA4 P48058 1/20 0.51
LCK P06239 1/20 0.45
PARP1 P09874 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
PLA2G10 O15496 1/20 0.43
MGAM O43451 1/20 0.43
PLA2G2A P14555 1/20 0.43
PLA2G5 P39877 1/20 0.43
PLA2G12A Q9BZM1 1/20 0.43
FASN P49327 1/20 0.41
POLB P06746 1/20 0.41
MAPT P10636 1/20 0.41
MAOB P27338 1/20 0.41
NOS1 P29475 1/20 0.41
GABRA1 P14867 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29235466 0.77 TP53 (0.46) LCKPARP1POLBGABRA1GABRA5
SCHEMBL7982949 0.77 GABRA5 (0.36) GRIA1GRIA2GRIA3GRIA4PARP1
SCHEMBL2468642 0.77 DAO (0.46) GABRA1GABRG2GABRB3GABRA5GABRA2
Lithium Ion SCHEMBL31177616 0.75 PARP1 (0.40) PARP1POLBGABRA5
SCHEMBL7983014 0.74 GABRA5 (0.46) LCKALDH1A1POLBMAPTGABRA1
SCHEMBL29235602 0.74 PARP1 (0.45) GRIA1GRIA2GRIA3GRIA4PARP1
SCHEMBL4763948 0.73 PARP1 (0.59) PARP1ALDH1A1POLBMAPTGABRA1
SCHEMBL30095396 0.73 PARP1 (0.59) PARP1ALDH1A1POLBMAPTGABRA1
SCHEMBL11557800 0.73 GRIA1 (0.48) GRIA1GRIA2GRIA3GRIA4PARP1
SCHEMBL8609965 0.71 CYP1A2 (0.57) GRIA1GRIA2GRIA3GRIA4PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed