SCHEMBL7982949

SCHEMBL7982949

O=c1[nH]c2ccc(I)cc2n2cncc12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA5 P31644 4/20 0.36
HTR1A P08908 2/20 0.35
HTR7 P34969 2/20 0.35
HTR6 P50406 2/20 0.35
PARP1 P09874 4/20 0.35
POLB P06746 1/20 0.34
CHEK1 O14757 1/20 0.34
CHEK2 O96017 1/20 0.34
CDK1 P06493 1/20 0.34
GSK3B P49841 1/20 0.34
PRKDC P78527 1/20 0.34
NOS1 P29475 1/20 0.33
DAO P14920 1/20 0.33
DRD2 P14416 1/20 0.33
GABRA1 P14867 2/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIA1 P42261 1/20 0.33
GRIA2 P42262 1/20 0.33
GRIA3 P42263 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468642 0.82 DAO (0.46) GABRA5DAOGABRA1GRIN2DGRIN3B
SCHEMBL7980241 0.82 DAO (0.46) GABRA5PARP1DAOGABRA1
SCHEMBL7983014 0.78 GABRA5 (0.46) GABRA5HTR1AHTR7HTR6POLB
SCHEMBL4763948 0.78 PARP1 (0.59) GABRA5PARP1POLBCHEK1CHEK2
SCHEMBL11997319 0.77 IDO1 (0.40) GABRA5PARP1CDK1GABRA1PBK
SCHEMBL7969955 0.77 GRIA1 (0.51) GABRA5PARP1POLBNOS1GABRA1
Lithium Ion SCHEMBL31177616 0.76 PARP1 (0.40) GABRA5PARP1POLBCHEK1CHEK2
SCHEMBL7969712 0.75 PGR (0.47) CHEK1GRIA1GRIA2GRIA3GRIA4
SCHEMBL31026820 0.74 PARP1 (0.49) HTR7HTR6PARP1
SCHEMBL4036186 0.73 PARP1 (0.42) GABRA5PARP1POLBCHEK1CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235740-B1 AUTOIMMUNE DISEASES; ANTIPROLIFERATION AGENTS BRISTOL-MYERS SQUIBB CO. 2001-05-22 US disclosed