SCHEMBL7970709

SCHEMBL7970709

CCc1cc(C#Cc2ccc(C3(OCc4ccccc4)CC3)c(CC)c2)ccc1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARB P10826 3/20 0.39
RARA P10276 2/20 0.39
RARG P13631 2/20 0.39
CYP26A1 O43174 1/20 0.39
CYP3A4 P08684 1/20 0.39
CRABP2 P29373 1/20 0.39
HNF4A P41235 1/20 0.35
RXRA P19793 3/20 0.35
SRD5A1 P18405 1/20 0.34
SRD5A2 P31213 1/20 0.34
MCL1 Q07820 1/20 0.34
LTB4R Q15722 1/20 0.34
LTB4R2 Q9NPC1 1/20 0.34
FOLH1 Q04609 1/20 0.34
CTSV O60911 1/20 0.34
CTSL P07711 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34
MRGPRX4 Q96LA9 2/20 0.33
ACACB O00763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980612 0.93 MCL1 (0.37) RARBRARARARGCYP26A1CYP3A4
SCHEMBL7987895 0.89 HNF4A (0.38) RARBRARARARGCYP26A1CYP3A4
SCHEMBL5735372 0.89 RARB (0.52) RARBRARARARGCYP26A1CYP3A4
SCHEMBL5737152 0.86 FFAR1 (0.48) RARBRARARARGCYP26A1CYP3A4
SCHEMBL6425907 0.83 ACACB (0.41) RARBRARARARGCYP26A1CYP3A4
SCHEMBL5735670 0.83 SMN1; SMN2 (0.45) RARBRARARARGCYP26A1CYP3A4
SCHEMBL5735734 0.82 GABRA1 (0.33) RARBRARARARGCYP26A1CYP3A4
SCHEMBL5737804 0.82 OPRM1 (0.34) ALDH1A1
SCHEMBL7980771 0.81 RARB (0.38) RARBRARARARGCYP26A1CYP3A4
SCHEMBL7984067 0.80 RARB (0.36) RARBRARARARGCYP26A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed