SCHEMBL7970840

SCHEMBL7970840

Nc1cc2c(=O)nc[nH]c2cn1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNP P00491 1/20 0.40
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.37
KDM4E B2RXH2 3/20 0.37
BLM P54132 2/20 0.37
APEX1 P27695 1/20 0.37
RECQL P46063 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
PRKCI P41743 1/20 0.35
PARP1 P09874 2/20 0.35
RXFP1 Q9HBX9 1/20 0.35
RAD52 P43351 1/20 0.34
PDE9A O76083 1/20 0.34
DYRK1A Q13627 1/20 0.33
ABL1 P00519 1/20 0.33
RIN1 Q13671 1/20 0.33
NOS3 P29474 2/20 0.32
NOS1 P29475 2/20 0.32
NOS2 P35228 2/20 0.32
MKNK1 Q9BUB5 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3319993 0.78 GABRP (0.42) PNPALDH1A1MAPTKDM4EBLM
SCHEMBL28490365 0.78 PARP1 (0.35) PNPALDH1A1MAPTKDM4EBLM
SCHEMBL7657497 0.78 UHRF1 (0.35) PNPALDH1A1MAPTPARP1PDE9A
SCHEMBL8934855 0.77 MAPT (0.53) PNPALDH1A1MAPTKDM4EBLM
SCHEMBL6360080 0.76 LCK (0.39) PNPALDH1A1MAPTKDM4EAPEX1
SCHEMBL6769664 0.75 CHEK1 (0.46) PDE9ACHEK1
SCHEMBL8700858 0.74 PARP1 (0.54) PNPALDH1A1MAPTKDM4EBLM
SCHEMBL6769400 0.74 PDE9A (0.38) PNPMAPTPDE9A
SCHEMBL6364136 0.74 GABRP (0.49) ALDH1A1MAPTKDM4EAPEX1PDE9A
SCHEMBL17769932 0.72 MAPT (0.57) PNPALDH1A1MAPTKDM4EBLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174889-B1 PROTEIN TYROSINE KINASE INHIBITORS RELATED TO BIOISOSTERES OF QUINOLINE AND QUINAZOLINE DERIVATIVES; ANTICARCINOGENIC AND -TUMOR AGENTS; PSORIASIS; RESTENOSIS; RHEUMATOID ARTHRITIS, AUTOIMMUNE DISEASE, ALLERGY, ASTHMA AND GRAFT REJECTION GLAXO WELLCOME INC. 2001-01-16 US claimed