SCHEMBL7970997

SCHEMBL7970997

O=C(NNC(=O)c1ccc(CNS(=O)(=O)c2ccccc2)cc1)c1ccccc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 1/20 0.69
GRIN1 Q05586 1/20 0.67
GRIN2A Q12879 1/20 0.67
GRIN2B Q13224 1/20 0.67
KEAP1 Q14145 1/20 0.65
MAPT P10636 3/20 0.63
NAMPT P43490 1/20 0.62
HTT P42858 3/20 0.60
HDAC8 Q9BY41 2/20 0.60
HDAC6 Q9UBN7 2/20 0.60
HDAC2 Q92769 1/20 0.60
KAT6A Q92794 1/20 0.59
CA12 O43570 1/20 0.59
CA1 P00915 1/20 0.59
CA2 P00918 1/20 0.59
CA9 Q16790 1/20 0.59
SMN1; SMN2 Q16637 4/20 0.58
LMNA P02545 3/20 0.58
HPGD P15428 2/20 0.58
OPRM1 P35372 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7973291 0.90 OPRK1 (0.65) CXCR4GRIN1GRIN2AGRIN2BMAPT
SCHEMBL19358860 0.88 CXCR4 (0.82) CXCR4KEAP1MAPTNAMPTHTT
SCHEMBL996398 0.86 KEAP1 (0.71) CXCR4KEAP1MAPTNAMPTHTT
SCHEMBL19358847 0.82 CXCR4 (0.77) CXCR4GRIN1GRIN2AGRIN2BKEAP1
SCHEMBL19358887 0.82 MAPT (0.82) CXCR4MAPTHTTCA12CA9
SCHEMBL19358855 0.82 CXCR4 (1.00) CXCR4KEAP1MAPTNAMPTHTT
SCHEMBL30254760 0.82 CXCR4 (0.78) CXCR4KEAP1MAPTHTTHDAC8
SCHEMBL15348918 0.81 GRIN1 (1.00) CXCR4GRIN1GRIN2AGRIN2BMAPT
SCHEMBL29557264 0.81 GRIN1 (1.00) CXCR4GRIN1GRIN2AGRIN2BMAPT
SCHEMBL1079531 0.81 NAMPT (0.67) CXCR4KEAP1MAPTNAMPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6271247-B1 BINDING TO NEUROPEPTIDE RECEPTORS ADIR ET COMPAGNIE (FR) 2001-08-07 US disclosed
US-6172108-B1 NEUROPEPTIDE Y RECEPTOR LIGANDS; TREATING PSYCHOLOGICAL, EATING, SLEEP, AND SEXUAL DISORDERS; HYPOTENSIVE, ANXIOLYTIC, ANTIDEPRESSANT, AND ANTIDIABETIC AGENTS ADIR ET COMPAGNIE (FR) 2001-01-09 US disclosed
EP-1010691-A2 Hydrazide derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2000-06-21 EP disclosed