SCHEMBL7971322

SCHEMBL7971322

CCCCCc1ccc(Oc2cccc(/C=C3\SC(=S)NC3=O)c2)cc1

nearest known ligand 0.70

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 8/20 0.70
MMP13 P45452 3/20 0.69
MMP3 P08254 2/20 0.69
GSK3B P49841 3/20 0.57
IDH1 O75874 1/20 0.54
AKR1B1 P15121 1/20 0.54
NAT1 P18440 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971324 1.00 ADAMTS5 (0.70) ADAMTS5MMP13MMP3GSK3BIDH1
SCHEMBL7969152 0.97 ADAMTS5 (0.72) ADAMTS5MMP13MMP3GSK3BIDH1
SCHEMBL7969157 0.97 ADAMTS5 (0.72) ADAMTS5MMP13MMP3GSK3BIDH1
SCHEMBL7972211 0.90 MMP3 (0.65) ADAMTS5MMP13MMP3NAT1
SCHEMBL7972208 0.90 MMP3 (0.65) ADAMTS5MMP13MMP3NAT1
SCHEMBL7958380 0.86 MMP3 (0.66) ADAMTS5MMP13MMP3NAT1
SCHEMBL7958378 0.86 MMP3 (0.66) ADAMTS5MMP13MMP3NAT1
SCHEMBL7971373 0.86 ADAMTS5 (0.76) ADAMTS5MMP13MMP3GSK3BIDH1
SCHEMBL7971376 0.86 ADAMTS5 (0.76) ADAMTS5MMP13MMP3GSK3BIDH1
SCHEMBL12685660 0.84 GSK3B (0.79) ADAMTS5MMP13MMP3GSK3BIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251928-B1 ADMINISTERING BENZYLIDENE RHODANINES WHICH ARE USEFUL AS AGENTS IN TREATING OR PREVENTING CONDITIONS ASSOCIATED WITH BETA-AMYLOID PEPTIDE IN A MAMMAL ELI LILLY AND COMPANY 2001-06-26 US disclosed
EP-0677517-A1 Treatment of Alzheimer's disease employing inhibitors of cathepsin D ELI LILLY AND COMPANY (US) 1995-10-18 EP disclosed