SCHEMBL7972159

SCHEMBL7972159

COc1c(C(=O)c2cccc3[nH]c(NS(=O)(=O)c4ccccc4)nc23)ccc(C(=O)N(C)c2ccc(C)cc2OCCCCCC(=O)N2CCN(C)CC2)c1N

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 1/20 0.34
AVPR1A P37288 1/20 0.34
HTR4 Q13639 4/20 0.32
CDK1 P06493 2/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32
CDK2 P24941 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
TDP1 Q9NUW8 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C19 P33261 1/20 0.31
AXL P30530 1/20 0.31
PDE3B Q13370 1/20 0.30
PDE3A Q14432 1/20 0.30
USP2 O75604 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473879 0.86 AVPR2 (0.34) AVPR2AVPR1ACDK1CDK4CCND1
SCHEMBL7480515 0.86 AVPR2 (0.35) AVPR2AVPR1AHTR4CDK1CDK4
SCHEMBL7961936 0.86 PARP1 (0.34) AVPR2AVPR1AHTR4CDK1CDK4
SCHEMBL7967392 0.84 AVPR2 (0.39) AVPR2AVPR1AMEN1KMT2A
Hydrochloric Acid SCHEMBL7970228 0.84 AVPR2 (0.33) AVPR2AVPR1A
Hydrochloric Acid SCHEMBL7970213 0.84 AVPR2 (0.38) AVPR2AVPR1AMEN1KMT2A
SCHEMBL7478475 0.81 CBX7 (0.38) AVPR2AVPR1AHTR4MEN1KMT2A
SCHEMBL7486482 0.80 RAB9A (0.35) AVPR2AVPR1ACDK1CDK4CCND1
SCHEMBL7340721 0.80 AVPR2 (0.39) AVPR2AVPR1ACDK1CDK4CCND1
SCHEMBL7781332 0.79 KMT2A (0.39) AVPR2AVPR1AHTR4MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6207693-B1 Benzamide derivatives having a vasopressin antagonistic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-03-27 US disclosed