SCHEMBL7972165

SCHEMBL7972165

CC(CCC(C#N)(c1ccccc1C(F)(F)F)C(C)C)N(C)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.50
EBP Q15125 3/20 0.50
KDM4E B2RXH2 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.37
MAOB P27338 5/20 0.35
MAOA P21397 4/20 0.35
CYP1A2 P05177 2/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
ADRA1A P35348 1/20 0.35
SNCA P37840 1/20 0.35
OPRK1 P41145 1/20 0.35
CYP2D6 P10635 1/20 0.35
PKM P14618 1/20 0.35
TSHR P16473 1/20 0.35
EPHX2 P34913 1/20 0.35
MAPK1 P28482 1/20 0.34
MLYCD O95822 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969369 0.91 SIGMAR1 (0.48) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7969794 0.89 SIGMAR1 (0.50) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7956095 0.89 SIGMAR1 (0.50) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7968611 0.89 ADRA2B (0.43) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7972515 0.89 SIGMAR1 (0.51) SIGMAR1EBPKDM4ECYP1A2ADRA2A
SCHEMBL7971289 0.88 SIGMAR1 (0.47) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7972078 0.87 SIGMAR1 (0.58) SIGMAR1EBPKDM4ECYP1A2ADRA2A
SCHEMBL7969207 0.87 SIGMAR1 (0.50) SIGMAR1EBPKDM4EL3MBTL1MAOB
SCHEMBL7956233 0.83 SIGMAR1 (0.73) SIGMAR1EBPL3MBTL1CYP1A2ADRA2A
SCHEMBL7968645 0.82 SIGMAR1 (0.58) SIGMAR1EBPKDM4ECYP1A2ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed