SCHEMBL7969369

SCHEMBL7969369

CC(CCC(C#N)(c1c(C(F)(F)F)cccc1C(F)(F)F)C(C)C)N(C)CCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.48
EBP Q15125 3/20 0.48
KDM4E B2RXH2 1/20 0.44
EPHX2 P34913 1/20 0.36
MAOB P27338 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP3A4 P08684 4/20 0.32
ABCB1 P08183 3/20 0.32
ABCC1 P33527 3/20 0.32
CYP2C19 P33261 2/20 0.32
MEN1 O00255 2/20 0.32
ABCB11 O95342 2/20 0.32
KMT2A Q03164 2/20 0.32
KCNH2 Q12809 2/20 0.32
TSHR P16473 2/20 0.32
LMNA P02545 2/20 0.32
SLC22A1 O15245 1/20 0.32
CACNA1F O60840 1/20 0.32
CHRM2 P08172 1/20 0.32
HTR1A P08908 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7972165 0.91 SIGMAR1 (0.50) SIGMAR1EBPKDM4EEPHX2MAOB
SCHEMBL7967090 0.89 ADRA2B (0.41) SIGMAR1EBPKDM4EEPHX2MAOB
SCHEMBL7972339 0.89 SIGMAR1 (0.46) SIGMAR1EBPKDM4EEPHX2L3MBTL1
SCHEMBL7968797 0.87 SIGMAR1 (0.50) SIGMAR1EBPKDM4EMAOBCYP3A4
SCHEMBL7972078 0.85 SIGMAR1 (0.58) SIGMAR1EBPKDM4ECYP3A4ABCB1
SCHEMBL7956537 0.85 SIGMAR1 (0.50) SIGMAR1EBPKDM4EMAOBCYP3A4
SCHEMBL7956095 0.85 SIGMAR1 (0.50) SIGMAR1EBPKDM4EMAOBL3MBTL1
SCHEMBL7972393 0.85 SIGMAR1 (0.50) SIGMAR1EBPKDM4EMAOBCYP3A4
SCHEMBL7972515 0.85 SIGMAR1 (0.51) SIGMAR1EBPKDM4ECYP3A4ABCB1
SCHEMBL7971841 0.84 SIGMAR1 (0.70) SIGMAR1EBPL3MBTL1CYP3A4ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265439-B1 Halogenated phenylacetonitrile alkylaminoalkylphenyl compounds as immunosuppressives G.D. SEARLE & CO. 2001-07-24 US disclosed
US-5451604-A Useful in organ transplant surgery G. D. SEARLE & CO. (US) 1995-09-19 US disclosed