SCHEMBL7972258

SCHEMBL7972258

BrCc1ccnc(-c2ccccc2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 2/20 0.53
LOXL2 Q9Y4K0 2/20 0.47
ALDH1A1 P00352 2/20 0.43
HTR1A P08908 1/20 0.43
HTR7 P34969 1/20 0.43
TRPA1 O75762 1/20 0.43
TSHR P16473 1/20 0.43
FFAR1 O14842 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PDCD1 Q15116 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
MIF P14174 1/20 0.40
AURKA O14965 1/20 0.40
HSP90AA1 P07900 1/20 0.40
PRKACA P17612 1/20 0.40
ADORA2A P29274 1/20 0.40
WNT3A P56704 1/20 0.40
PIM1 P11309 1/20 0.40
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29871243 0.83 CCR1 (0.42) LOXL2ALDH1A1TRPA1TSHRPDCD1
SCHEMBL1259178 0.83 CCR1 (0.42) LOXL2ALDH1A1TRPA1TSHRPDCD1
SCHEMBL2956020 0.81 LOXL2 (0.43) LOXL2ALDH1A1HTR1ACYP11B1CYP11B2
Bromide SCHEMBL16739305 0.81 CCR1 (0.41) LOXL2ALDH1A1TRPA1TSHR
SCHEMBL7037544 0.81 KDM4E (0.54) ALDH1A1TRPA1TSHRHSP90AA1PIM1
SCHEMBL5991845 0.81 LOXL2 (0.70) ASIC3LOXL2HTR1AHTR7AURKA
SCHEMBL995901 0.81 ASIC3 (0.53) ASIC3LOXL2HTR1AHTR7TSHR
SCHEMBL4116786 0.81 ASIC3 (0.53) ASIC3LOXL2ALDH1A1HTR1AHTR7
SCHEMBL10434579 0.81 ASIC3 (0.53) ASIC3LOXL2HTR1AHTR7FFAR1
SCHEMBL10271516 0.81 ASIC3 (0.53) ASIC3LOXL2ALDH1A1HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118165038-A Cyclic metal ruthenium nitrosyl complex, preparation method and application as NO release photosensitizer 中南民族大学 2024-06-11 CN claimed
CN-118165038-A Cyclic metal ruthenium nitrosyl complex, preparation method and application as NO release photosensitizer 中南民族大学 2024-06-11 CN disclosed
EP-3750890-A1 ALKOXYBENZO-FIVE-MEMBERED (SIX-MEMBERED) HETEROCYCLIC AMINE COMPOUND AND PHARMACEUTICAL USE THEREOF Fudan University (CN) 2020-12-16 EP disclosed
WO-2019154047-A1 ALKOXYBENZO-FIVE-MEMBERED (SIX-MEMBERED) HETEROCYCLIC AMINE COMPOUND AND PHARMACEUTICAL USE THEREOF 复旦大学 2019-08-15 WO disclosed
US-6281359-B1 PSYCHOLOGICAL DISORDERS NEUROGEN CORPORATION 2001-08-28 US disclosed
US-6221871-B1 TREATING SCHIZOPHRENIA, DEPRESSION OR PARKINSON'S DISEASE NEUROGEN CORPORATION 2001-04-24 US disclosed
US-5912350-A Certain aminomethyl biphenyl, aminomethyl phenyl pyridine and aminomethyl phenyl pyrimidine derivatives; novel dopamine receptor subtype selective ligands NEUROGEN CORPORATION (US) 1999-06-15 US disclosed
US-5677454-A DIAGNOSIS, THERAPY OF SCHIZOPHRENIA, DEPRESSION, PARKINSONISM NEUROGEN CORPORATION (US) 1997-10-14 US disclosed
EP-0793662-A1 AMINOMETHYL ARYL COMPOUNDS; DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS NEUROGEN CORPORATION (US) 1997-09-10 EP disclosed
US-5594141-A ANTIPSYCHOTIC AND ANTIDEPRESSANT AGENTS; PARKINSON'S DISEASE NEUROGEN CORPORATION (US) 1997-01-14 US disclosed
WO-1996016058-A1 AMINOMETHYL ARYL COMPOUNDS; DOPAMINE RECEPTOR SUBTYPE SELECTIVE LIGANDS NEUROGEN CORPORATION (US) 1996-05-30 WO disclosed