Nifenalol

Nifenalol

SCHEMBL79725

CC(C)NCC(O)c1ccc([N+](=O)[O-])cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.66
ALDH1A1 P00352 3/20 0.62
NPSR1 Q6W5P4 1/20 0.62
ADRB2 P07550 6/20 0.57
ADRB1 P08588 6/20 0.57
ADRB3 P13945 5/20 0.57
MEN1 O00255 5/20 0.55
KMT2A Q03164 5/20 0.55
LMNA P02545 3/20 0.54
KDM4E B2RXH2 3/20 0.54
BLM P54132 2/20 0.52
GLA P06280 1/20 0.52
MAPT P10636 3/20 0.51
TSHR P16473 3/20 0.51
MTOR P42345 2/20 0.51
MAPK1 P28482 2/20 0.51
HSD17B10 Q99714 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
CYP1A2 P05177 2/20 0.51
HIF1A Q16665 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Nifenalol SCHEMBL6510064 1.00 NPC1 (0.66) NPC1ALDH1A1NPSR1ADRB2ADRB1
Nifenalol SCHEMBL9118298 0.98 NPC1 (0.64) NPC1ALDH1A1NPSR1ADRB2ADRB1
Nifenalol SCHEMBL28286362 0.97 NPC1 (0.62) NPC1ALDH1A1NPSR1ADRB2ADRB1
Sotalol SCHEMBL10898829 0.87 ADRB3 (0.78) NPC1ALDH1A1NPSR1ADRB2ADRB1
SCHEMBL4627256 0.86 NPC1 (0.61) NPC1ALDH1A1NPSR1ADRB2ADRB1
SCHEMBL2299495 0.84 MEN1 (0.62) NPC1ALDH1A1NPSR1MEN1KMT2A
SCHEMBL2292066 0.84 MEN1 (0.62) NPC1ALDH1A1NPSR1MEN1KMT2A
SCHEMBL28727682 0.84 MEN1 (0.62) NPC1ALDH1A1NPSR1MEN1KMT2A
SCHEMBL2292479 0.84 MEN1 (0.62) NPC1ALDH1A1NPSR1MEN1KMT2A
SCHEMBL2295250 0.84 MEN1 (0.62) NPC1ALDH1A1NPSR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1717 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119233997-A Tetrahedral antibodies 生物分子控股有限责任公司 2024-12-31 CN claimed
EP-4463485-A2 TETRAHEDRAL ANTIBODIES Biomolecular Holdings LLC (US) 2024-11-20 EP claimed
CN-116680820-A Optimization design method for deep groove ball bearing fatigue life-prolonging structure 南昌航空大学 2023-09-01 CN claimed
WO-2023137387-A2 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-20 WO claimed
WO-2023137373-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-20 WO claimed
US-20230220115-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-13 US claimed
US-20230220116-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2023-07-13 US claimed
EP-4178615-A1 TETRAHEDRAL ANTIBODIES Biomolecular Holdings LLC (US) 2023-05-17 EP claimed
US-11225490-B2 Prodrugs of secondary amine compounds ALKERMES PHARMA IRELAND LIMITED (IE) 2022-01-18 US claimed
WO-2022011358-A1 TETRAHEDRAL ANTIBODIES BIOMOLECULAR HOLDINGS LLC (US) 2022-01-13 WO claimed
EP-0152379-A2 Process for preparing pharmaceutical compositions containing unilamellar liposomes CIBA-GEIGY AG (CH) 1985-08-21 EP claimed
EP-0073819-A4 NASAL ADMINISTRATION OF BETA-BLOCKERS AND DOSAGE FORMS THEREFOR. UNIV KENTUCKY RES FOUND (US) 1984-11-16 EP claimed
US-4468391-A Combination of β-adrenoceptor antagonists and anxiolytic agents AYERST, MCKENNA & HARRISON, INC. (CA) 1984-08-28 US claimed
US-4428883-A NASAL OINTMENTS OR GELS THE UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1984-01-31 US claimed
EP-0098113-A1 A combination of beta-adrenoceptor antagonists and anxiolytic agents AYERST, MCKENNA AND HARRISON INC. (CA) 1984-01-11 EP claimed
EP-0073819-A1 NASAL ADMINISTRATION OF BETA-BLOCKERS AND DOSAGE FORMS THEREFOR. UNIV KENTUCKY RES FOUND (US) 1983-03-16 EP claimed
WO-1982003009-A1 NASAL ADMINISTRATION OF BETA-BLOCKERS AND DOSAGE FORMS THEREFOR UNIV KENTUCKY RES FOUND (US) 1982-09-16 WO claimed
US-4303637-A Medication indicated for ocular hypertension ALZA CORPORATION (US) 1981-12-01 US claimed
EP-0037622-A2 Drug delivery insert for controlled ocular therapy ALZA CORPORATION (US) 1981-10-14 EP claimed
US-4281654-A Drug delivery system for controlled ocular therapy ALZA CORPORATION (US) 1981-08-04 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230220115-A1 TETRAHEDRAL ANTIBODIES FCGR3B, FCGR2A, FCGR1A NPC1 3426/4885ALDH1A1 4781/4885NPSR1 331/4885
US-20230220116-A1 TETRAHEDRAL ANTIBODIES FCGR3B, FCGR2A, FCGR1A NPC1 3426/4885ALDH1A1 4781/4885NPSR1 331/4885
US-11225490-B2 Prodrugs of secondary amine compounds HNMT, MAOB, UGT1A1 NPC1 220/4885ALDH1A1 288/4885NPSR1 58/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.