SCHEMBL7973086

SCHEMBL7973086

CCN(CC)C(=O)Oc1c(-c2ccc(Cn3cccn3)cc2)n[nH]c1-c1nc2cc3c(cc2[nH]1)CNC3

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 1/20 0.33
HDAC1 Q13547 2/20 0.32
HDAC6 Q9UBN7 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC2 Q92769 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
KLKB1 P03952 2/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.31
KDR P35968 1/20 0.31
CXCR3 P49682 2/20 0.31
BRPF1 P55201 1/20 0.30
CA12 O43570 1/20 0.30
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30
CA9 Q16790 1/20 0.30
FGFR1 P11362 1/20 0.30
FLT1 P17948 1/20 0.30
KDM4E B2RXH2 1/20 0.30
AURKA O14965 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140005 0.87 PTGDR2 (0.33) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL7960749 0.85 HDAC3 (0.43) GRK6HDAC1HDAC6HDAC3HDAC2
SCHEMBL7973068 0.81 CHEK2 (0.39) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL7970984 0.80 SYK (0.32)
SCHEMBL7973410 0.74 PTGDR2 (0.36) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL20307807 0.73 KMT2A (0.34) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL10140040 0.73 CHEK2 (0.34)
SCHEMBL7975823 0.72 HDAC3 (0.43) HDAC1HDAC6HDAC3HDAC2HDAC8
SCHEMBL10140128 0.71 F10 (0.34) HDAC1HDAC6KLKB1PTGDR2BRPF1
SCHEMBL7972878 0.71 HPSE (0.38) KDRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed