SCHEMBL7972878

SCHEMBL7972878

CNC(=O)Oc1c(-c2ccc(C)cc2)n[nH]c1-c1nc2cc3c(cc2[nH]1)CNC3

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPSE Q9Y251 2/20 0.38
CHEK2 O96017 6/20 0.36
EGFR P00533 1/20 0.35
BRD4 O60885 1/20 0.35
RHEB Q15382 1/20 0.33
CDK4 P11802 1/20 0.33
CCNA2 P20248 1/20 0.33
CCND1 P24385 1/20 0.33
CDK2 P24941 1/20 0.33
CCND3 P30281 1/20 0.33
ALDH1A1 P00352 3/20 0.33
MAPT P10636 3/20 0.33
KDM4E B2RXH2 2/20 0.33
POLB P06746 2/20 0.33
HPGD P15428 2/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
KMT2A Q03164 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CASP3 P42574 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7975606 0.85 BRD4 (0.37) CHEK2BRD4NPC1RAB9ASMN1; SMN2
SCHEMBL7960176 0.84 BRD4 (0.36) CHEK2BRD4NPC1RAB9ASMN1; SMN2
SCHEMBL7975112 0.80 F9 (0.47) HPSECHEK2BRD4ALDH1A1MAPT
SCHEMBL7973068 0.79 CHEK2 (0.39) HPSECHEK2RHEBCDK4CCNA2
SCHEMBL20307729 0.76 F9 (0.40) HPSECHEK2CDK4CCNA2CCND1
SCHEMBL7969308 0.76 TSPO (0.37) CHEK2EGFRBRD4KDR
SCHEMBL7980011 0.73 CHEK2 (0.38) HPSECHEK2EGFRBRD4ALDH1A1
SCHEMBL7970984 0.72 SYK (0.32)
SCHEMBL7977818 0.72 F9 (0.48) CDK4CCNA2CCND1CDK2CCND3
SCHEMBL7960749 0.71 HDAC3 (0.43) CDK4CDK2KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed