SCHEMBL7973068

SCHEMBL7973068

CCN(CC)C(=O)Oc1c(-c2ccc(-c3ccc(C(=O)NC)cc3)cc2)n[nH]c1-c1nc2cc3c(cc2[nH]1)CNC3

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.39
CHEK1 O14757 1/20 0.38
CDK4 P11802 1/20 0.37
CCNA2 P20248 1/20 0.37
CCND1 P24385 1/20 0.37
CDK2 P24941 1/20 0.37
CCND3 P30281 1/20 0.37
FLT3 P36888 2/20 0.34
HDAC6 Q9UBN7 4/20 0.34
PRKAG1 P54619 1/20 0.33
PRKAA2 P54646 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
SYK P43405 1/20 0.33
ITK Q08881 1/20 0.33
HDAC3 O15379 3/20 0.33
HDAC1 Q13547 3/20 0.33
HDAC8 Q9BY41 3/20 0.33
HDAC2 Q92769 2/20 0.33
HPSE Q9Y251 1/20 0.33
PRSS12 P56730 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10140006 0.85 CHEK2 (0.38) CHEK2CDK4CCNA2CCND1CDK2
SCHEMBL7970984 0.82 SYK (0.32) SYKITK
SCHEMBL7960749 0.81 HDAC3 (0.43) CHEK1CDK4CDK2FLT3HDAC6
SCHEMBL7973086 0.81 GRK6 (0.33) HDAC6HDAC3HDAC1HDAC8HDAC2
SCHEMBL7972878 0.79 HPSE (0.38) CHEK2CDK4CCNA2CCND1CDK2
SCHEMBL10172564 0.77 MAPT (0.37) HDAC6HDAC1HPSE
SCHEMBL7960714 0.76 CHEK2 (0.39) CHEK2
SCHEMBL10140040 0.74 CHEK2 (0.34) CHEK2
SCHEMBL7969308 0.73 TSPO (0.37) CHEK2SYKITK
SCHEMBL7975606 0.72 BRD4 (0.37) CHEK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009143039-A2 HETEROCYCLIC COMPOUNDS AS FACTOR IXA INHIBITORS SCHERING CORPORATION (US) 2009-11-26 WO disclosed