SCHEMBL7974035

SCHEMBL7974035

Fc1ccc(-c2nnc3cc(N4CC=CCC4)c(Cl)nn23)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 3/20 0.35
HSD17B10 Q99714 2/20 0.34
PIM1 P11309 2/20 0.34
MAPK14 Q16539 1/20 0.34
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32
BACE1 P56817 1/20 0.32
AKT1 P31749 1/20 0.32
DPP4 P27487 1/20 0.32
F2RL1 P55085 3/20 0.32
HSD11B1 P28845 2/20 0.32
MAP4K4 O95819 2/20 0.31
EGFR P00533 2/20 0.31
CSNK1D P48730 2/20 0.31
PRKD2 Q9BZL6 2/20 0.31
MAPK9 P45984 1/20 0.31
MINK1 Q8N4C8 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2655376 0.87 HSD17B10 (0.43) P2RX7HSD17B10PIM1MAPK14BCHE
SCHEMBL7987232 0.80 KMT2A (0.41) HSD17B10PIM1DPP4PRKD2KDM4E
SCHEMBL7991356 0.76 GABRG2 (0.57)
SCHEMBL7984270 0.75 BCHE (0.39) HSD17B10BCHEKDM4EALDH1A1POLB
SCHEMBL6773500 0.69 MAPK14 (0.39) P2RX7HSD17B10PIM1MAPK14HSD11B1
SCHEMBL7987387 0.66 NPC1 (0.40) BCHEACHEBACE1EGFRKDM4E
SCHEMBL7987392 0.66 NPC1 (0.40) BCHEACHEBACE1EGFRKDM4E
SCHEMBL6775681 0.66 HSD11B1 (0.43) HSD11B1POLB
SCHEMBL6775795 0.63 DCTPP1 (0.45) HSD11B1ALDH1A1POLB
SCHEMBL7972521 0.63 BCHE (0.42) HSD17B10BCHEKDM4EALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6319924-B1 FOR THERAPY OF DELETERIOUS MENTAL STATES MERCK SHARP & DOHME LTD. (GB) 2001-11-20 US disclosed