SCHEMBL7974089

SCHEMBL7974089

O[C@H](COc1ccc2c(c1)OCO2)CN1CCC(c2noc3cc(F)ccc23)CC1

nearest known ligand 0.69

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.68
DRD2 P14416 4/20 0.68
HTR1A P08908 1/20 0.68
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57
POLB P06746 1/20 0.56
DRD3 P35462 2/20 0.53
MEN1 O00255 1/20 0.53
KMT2A Q03164 1/20 0.53
ACHE P22303 2/20 0.52
SLC6A4 P31645 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7974099 1.00 HTR2A (0.68) HTR2ADRD2HTR1AALDH1A1MAPT
SCHEMBL1545448 0.86 HTR2A (0.77) HTR2ADRD2HTR1ADRD3ACHE
SCHEMBL5368375 0.84 HTR2A (0.72) HTR2ADRD2HTR1ADRD3ACHE
SCHEMBL5368366 0.84 HTR2A (0.72) HTR2ADRD2HTR1ADRD3ACHE
SCHEMBL7496035 0.82 HTR2A (0.69) HTR2ADRD2HTR1ADRD3ACHE
Hydrochloric Acid SCHEMBL1545656 0.81 ACHE (0.69) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL15703012 0.81 KCNH2 (0.74) HTR2ADRD2HTR1AALDH1A1MAPT
SCHEMBL7977213 0.80 HTR2A (0.60) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL1545018 0.80 DRD2 (0.72) HTR2ADRD2HTR1AACHESLC6A4
SCHEMBL20512970 0.80 DRD2 (1.00) HTR2ADRD2HTR1ADRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001017993-A1 ALKYLPIPERIDI NYLBENZO [D] ISOXAZOLE DERIVATIVES HAVING PSYCHOTROPIC ACTIVITY, PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME, AND A PROCESS FOR THE PREPARATION OF THE ACTIVE INGREDIENT EGIS Gyógyszergyár Rt. (HU) 2001-03-15 WO disclosed