SCHEMBL7976436

SCHEMBL7976436

CCOC(=O)N1CCC(SC(c2ccccc2)c2ccccc2)CC1

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.58
GAA P10253 2/20 0.56
ALDH1A1 P00352 4/20 0.52
KDM4E B2RXH2 3/20 0.52
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
BRD4 O60885 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.51
MAPT P10636 1/20 0.49
HPGD P15428 1/20 0.49
CHRM2 P08172 1/20 0.48
CHRM5 P08912 1/20 0.48
CHRM3 P20309 1/20 0.48
NOS2 P35228 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9216384 0.82 KMT2A (0.53) TSHRALDH1A1KDM4EKMT2ABRD4
SCHEMBL9353361 0.82 KDM4E (0.46) ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL9352843 0.81 ALDH1A1 (0.45) ALDH1A1KDM4EKMT2AMEN1L3MBTL1
SCHEMBL14198379 0.81 TSHR (0.63) TSHRGAAALDH1A1KDM4EKMT2A
SCHEMBL9353421 0.80 HTR4 (0.47) ALDH1A1KDM4ECHRM2CHRM5CHRM3
SCHEMBL4255064 0.77 TSHR (0.59) TSHRGAAALDH1A1KDM4EKMT2A
SCHEMBL6980957 0.77 KMT2A (0.63) TSHRGAAALDH1A1KDM4EKMT2A
SCHEMBL20618720 0.75 TSHR (0.60) TSHRGAAALDH1A1KDM4EKMT2A
Hydrochloric Acid SCHEMBL9353101 0.75 HSP90AA1 (0.39) GAAKDM4E
SCHEMBL7965918 0.74 CHRM2 (0.51) GAAKDM4ECHRM2CHRM5CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000034437-A2 INHIBITORS OF PRENYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 2000-06-15 WO claimed
US-6255323-B1 Cyanoguanidine compounds SHIONOGI BIORESEARCH CORP. 2001-07-03 US disclosed
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO disclosed
EP-0399414-B1 Piperidine derivative, method for preparation thereof, and a pharmaceutical composition comprising the same HOKURIKU PHARMACEUTICAL (JP) 1994-09-21 EP disclosed
US-5153207-A Antihistamine and antiallergic agent HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1992-10-06 US disclosed
EP-0399414-A1 Piperidine derivative, method for preparation thereof, and a pharmaceutical composition comprising the same HOKURIKU PHARMACEUTICAL CO., LTD. (JP) 1990-11-28 EP disclosed