SCHEMBL7976689

SCHEMBL7976689

COc1ccc(C#N)cc1-c1ccc(OC(C)C(O)CCc2cccnc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
PTAFR P25105 9/20 0.40
SCN9A Q15858 1/20 0.40
PDE5A O76074 1/20 0.39
KDM1A O60341 2/20 0.38
CHEK1 O14757 1/20 0.38
CD274 Q9NZQ7 1/20 0.38
ALPL P05186 1/20 0.38
KDM4E B2RXH2 2/20 0.37
NPC1 O15118 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GAA P10253 1/20 0.37
HPGD P15428 1/20 0.37
CTSA P10619 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976694 1.00 CYP19A1 (0.41) CYP19A1CYP11B1CYP11B2PTAFRSCN9A
SCHEMBL8019943 1.00 CYP19A1 (0.41) CYP19A1CYP11B1CYP11B2PTAFRSCN9A
SCHEMBL7966320 0.88 CYP11B1 (0.40) CYP19A1CYP11B1CYP11B2PTAFRSCN9A
SCHEMBL7966319 0.88 CYP11B1 (0.40) CYP19A1CYP11B1CYP11B2PTAFRSCN9A
SCHEMBL7978652 0.87 CYP11B2 (0.43) CYP19A1CYP11B1CYP11B2PTAFR
SCHEMBL7978653 0.87 CYP11B2 (0.43) CYP19A1CYP11B1CYP11B2PTAFR
SCHEMBL7822506 0.84 CYP11B2 (0.38) CYP19A1CYP11B1CYP11B2PTAFRHPGD
SCHEMBL7822509 0.84 CYP11B2 (0.38) CYP19A1CYP11B1CYP11B2PTAFRHPGD
SCHEMBL7980395 0.84 MMP12 (0.47) CYP19A1CYP11B1CYP11B2PTAFRKDM4E
SCHEMBL7980127 0.84 MMP12 (0.47) CYP19A1CYP11B1CYP11B2PTAFRKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6300352-B1 FOR THERAPY OF ASTHMA ASTRAZENECA AB (SE) 2001-10-09 US claimed
EP-0971892-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Astra Pharmaceuticals Limited (GB) 2000-01-19 EP claimed
WO-1998042670-A1 NOVEL PYRIDINE DERIVATIVES AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM ASTRA PHARMACEUTICALS LTD. (GB) 1998-10-01 WO claimed
US-6300352-B1 FOR THERAPY OF ASTHMA ASTRAZENECA AB (SE) 2001-10-09 US disclosed