SCHEMBL7976803

SCHEMBL7976803

CC(CN(C)C)Cn1cc(-c2cncc(-c3ccsc3)c2)c2ncccc21

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.75
FLT1 P17948 4/20 0.75
FLT4 P35916 4/20 0.75
CYP2A6 P11509 5/20 0.39
MAOB P27338 1/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2B6 P20813 1/20 0.34
CYP2C19 P33261 1/20 0.34
PRKACA P17612 1/20 0.34
PRKACG P22612 1/20 0.34
PRKACB P22694 1/20 0.34
DYRK1A Q13627 2/20 0.33
GAK O14976 1/20 0.33
KCNH2 Q12809 1/20 0.33
CHEK2 O96017 1/20 0.32
CLK3 P49761 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7986720 0.88 KDR (0.59) KDRFLT1FLT4CYP3A4PRKACA
SCHEMBL7547755 0.86 KDR (1.00) KDRFLT1FLT4CYP2A6PRKACA
SCHEMBL7551380 0.85 KDR (0.54) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7555413 0.83 KDR (0.52) KDRFLT1FLT4PRKACAPRKACG
SCHEMBL7549028 0.83 KDR (0.52) KDRFLT1FLT4MAOBCYP3A4
SCHEMBL7508695 0.83 KDR (0.74) KDRFLT1FLT4CYP2A6MAOB
SCHEMBL7987137 0.83 KDR (0.74) KDRFLT1FLT4CYP2A6PRKACA
SCHEMBL7547036 0.82 FLT1 (0.51) KDRFLT1FLT4MAOBCYP3A4
SCHEMBL7988018 0.80 KDR (0.78) KDRFLT1FLT4CYP2A6PRKACA
SCHEMBL7976429 0.80 KDR (0.78) KDRFLT1FLT4CYP2A6PRKACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed