SCHEMBL7976982

SCHEMBL7976982

O=c1[nH]nc(O)c2c1Cc1c(Cl)cc(Cl)cc1N2

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.35
HTR6 P50406 1/20 0.32
PARP1 P09874 1/20 0.31
DNMT1 P26358 1/20 0.31
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
AHR P35869 2/20 0.30
CMA1 P23946 1/20 0.30
GSK3A P49840 1/20 0.30
GSK3B P49841 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978816 0.81 AHR (0.51) CES1AHRCMA1
SCHEMBL7478045 0.80 CES1 (0.40) CES1HTR6DNMT1ALDH1A1TP53
SCHEMBL7478394 0.68 OPRM1 (0.38) ALDH1A1MAPT
SCHEMBL7479024 0.68 RXRA (0.42) HTR6ALDH1A1MAPT
SCHEMBL7483973 0.62 AHR (0.45) PARP1AHRCMA1
SCHEMBL8873506 0.62 ALDH1A1 (0.37) CES1HTR6DNMT1ALDH1A1MAPT
SCHEMBL18623469 0.60 GRIN2D (0.46) ALDH1A1GSK3BCDK5
SCHEMBL8871800 0.60 CES1 (0.49) CES1HTR6DNMT1ALDH1A1TP53
SCHEMBL8874319 0.59 CES1 (0.47) CES1HTR6DNMT1ALDH1A1AHR
SCHEMBL8874292 0.59 CES1 (0.52) CES1HTR6PARP1DNMT1AHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6214826-B1 NERVOUS SYSTEM DISORDERS ZENECA LIMITED (GB) 2001-04-10 US claimed