SCHEMBL7976983

SCHEMBL7976983

CCOc1noc2c1C(NCc1ccccc1)CCC2

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.45
CHRM2 P08172 2/20 0.38
CHRM4 P08173 2/20 0.38
CHRM5 P08912 2/20 0.38
CHRM1 P11229 2/20 0.38
CHRM3 P20309 2/20 0.38
KMT2A Q03164 2/20 0.37
LMNA P02545 1/20 0.37
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
OPRK1 P41145 1/20 0.36
NPC1 O15118 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724638 0.81 HTR2A (0.35) KDM4ECHRM2CHRM4CHRM5CHRM1
SCHEMBL5725539 0.79 HTR2C (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5725534 0.79 HTR2C (0.47) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5724839 0.79 CHRM3 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5725074 0.79 CHRM3 (0.45) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL5726347 0.79 CHRM2 (0.32) KDM4ECHRM2CHRM4CHRM5CHRM1
SCHEMBL5726344 0.79 CHRM2 (0.32) KDM4ECHRM2CHRM4CHRM5CHRM1
Bromide SCHEMBL5726761 0.79 LMNA (0.44) KDM4EKMT2ALMNAALDH1A1NPC1
Bromide SCHEMBL5726756 0.79 LMNA (0.44) KDM4EKMT2ALMNAALDH1A1NPC1
SCHEMBL5725224 0.78 CHRM2 (0.32) CHRM2CHRM4CHRM5CHRM1CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed