SCHEMBL5725539

SCHEMBL5725539

CN[C@@H]1CCCc2onc(OCc3ccccc3)c21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 5/20 0.47
HTR2A P28223 4/20 0.47
CHRM2 P08172 1/20 0.46
CHRM4 P08173 1/20 0.46
CHRM5 P08912 1/20 0.46
CHRM1 P11229 1/20 0.46
CHRM3 P20309 1/20 0.46
SLC6A4 P31645 5/20 0.37
CNR2 P34972 3/20 0.35
CNR1 P21554 2/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
HTR1A P08908 1/20 0.34
SLC6A2 P23975 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5725534 1.00 HTR2C (0.47) HTR2CHTR2ACHRM2CHRM4CHRM5
SCHEMBL5724839 0.81 CHRM3 (0.45) HTR2CHTR2ACHRM2CHRM4CHRM5
SCHEMBL8350478 0.79 DHODH (0.37) LMNAKMT2A
SCHEMBL7976973 0.79 DHODH (0.37) LMNAKMT2A
SCHEMBL7976983 0.79 KDM4E (0.45) HTR2CHTR2ACHRM2CHRM4CHRM5
SCHEMBL5725434 0.78 SIGMAR1 (0.40) HTR2CHTR2ACHRM2CHRM4CHRM5
SCHEMBL5725047 0.77 ENPP3 (0.34) CA2CA9
SCHEMBL8351808 0.75 L3MBTL1 (0.37) L3MBTL1LMNAKMT2A
SCHEMBL8351806 0.75 L3MBTL1 (0.37) L3MBTL1LMNAKMT2A
SCHEMBL7983154 0.73 KDM4E (0.35) L3MBTL1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0812318-B1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS LUNDBECK & CO AS H (DK) 2006-02-08 EP disclosed
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed