SCHEMBL7976998

SCHEMBL7976998

COC(=O)CNC(=O)C(CCCCNC(C)=N)NC(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.49
CTSS P25774 6/20 0.49
CA1 P00915 3/20 0.45
CA2 P00918 3/20 0.45
CAPN1 P07384 1/20 0.43
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
CXCR3 P49682 2/20 0.42
HDAC6 Q9UBN7 1/20 0.42
SIRT5 Q9NXA8 1/20 0.41
MEN1 O00255 1/20 0.40
GAA P10253 1/20 0.40
KMT2A Q03164 1/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
ITGB3 P05106 1/20 0.39
ITGA2B P08514 1/20 0.39
JAK3 P52333 1/20 0.39
BTK Q06187 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13702236 0.90 CTSK (0.53) CTSKCTSSCA1CA2CAPN1
SCHEMBL30312666 0.90 CTSK (0.53) CTSKCTSSCA1CA2CAPN1
SCHEMBL7700364 0.84 MEN1 (0.51) CTSKCTSSCA1CA2CAPN1
SCHEMBL7974820 0.84 MEN1 (0.51) CTSKCTSSCA1CA2CAPN1
SCHEMBL7977002 0.83 CTSK (0.46) CTSKCTSSCA1CA2CAPN1
SCHEMBL7963473 0.81 CTSS (0.45) CTSKCTSSCA1CA2CAPN1
SCHEMBL16924919 0.81 CTSK (0.51) CTSKCTSSCA1CA2CAPN1
SCHEMBL30312609 0.80 CTSS (0.56) CTSKCTSSCA1CA2CAPN1
SCHEMBL13702232 0.80 CTSS (0.56) CTSKCTSSCA1CA2CAPN1
SCHEMBL10144100 0.80 CTSS (0.51) CTSKCTSSCA2CAPN1HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001005748-A1 OLIGOMERIC AMINO ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS MONSANTO COMPANY (US) 2001-01-25 WO disclosed