SCHEMBL7977002

SCHEMBL7977002

COC(=O)CNC(=O)C(CCCCNCC=N)NC(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSK P43235 7/20 0.46
CTSS P25774 6/20 0.46
HDAC4 P56524 3/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC6 Q9UBN7 1/20 0.42
JAK3 P52333 1/20 0.42
BTK Q06187 1/20 0.42
F10 P00742 1/20 0.40
CAPN1 P07384 1/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
CXCR3 P49682 1/20 0.38
CTSL P07711 1/20 0.38
CTSB P07858 1/20 0.38
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
SIRT5 Q9NXA8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13702236 0.85 CTSK (0.53) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL30312666 0.85 CTSK (0.53) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL7973800 0.84 CTSK (0.41) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL7974823 0.83 ALDH1A1 (0.47) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL7976998 0.83 CTSK (0.49) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL7974856 0.82 CTSK (0.43) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL12081854 0.79 JAK3 (0.68) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL16383457 0.76 CTSS (0.52) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL16924919 0.75 CTSK (0.51) CTSKCTSSHDAC4HDAC1HDAC6
SCHEMBL7977282 0.75 TDP1 (0.40) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001005748-A1 OLIGOMERIC AMINO ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS MONSANTO COMPANY (US) 2001-01-25 WO disclosed