SCHEMBL7977700

SCHEMBL7977700

Nc1cccc(-c2cc3c(Br)cccc3c(N)n2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.49
MEN1 O00255 4/20 0.49
MAPT P10636 4/20 0.49
KDM4E B2RXH2 3/20 0.49
KMT2A Q03164 3/20 0.49
LMNA P02545 3/20 0.49
HPGD P15428 3/20 0.49
GLA P06280 1/20 0.45
RAB9A P51151 3/20 0.42
NPC1 O15118 2/20 0.42
TSHR P16473 1/20 0.42
RECQL P46063 1/20 0.42
METAP2 P50579 1/20 0.41
POLB P06746 1/20 0.40
GFER P55789 1/20 0.40
MAOA P21397 1/20 0.39
PDPK1 O15530 1/20 0.39
AURKA O14965 1/20 0.39
MAP4K4 O95819 3/20 0.38
NFKB1 P19838 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978412 0.79 ALDH1A1 (0.57) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL17873008 0.71 BACE1 (0.42) ALDH1A1KDM4EMAP4K4BACE1
SCHEMBL12072247 0.68 ACHE (0.49) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL6733442 0.67 MEN1 (0.89) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL14389682 0.67 MEN1 (0.70) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL25735690 0.67 TSHR (0.68) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL15690753 0.66 MEN1 (0.93) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL15684033 0.66 MEN1 (0.73) ALDH1A1MEN1MAPTKDM4EKMT2A
SCHEMBL2261782 0.66 XDH (0.52) IKBKB
SCHEMBL30165334 0.66 MEN1 (0.57) ALDH1A1MEN1MAPTKDM4EKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed