SCHEMBL7977980

SCHEMBL7977980

CCc1ncnc(NC2COC(c3ccc(C)cc3)OC2)c1Cl

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.33
LMNA P02545 1/20 0.33
ADORA3 P0DMS8 3/20 0.31
ADORA2A P29274 3/20 0.31
ADORA1 P30542 3/20 0.31
ADORA2B P29275 2/20 0.31
GRM1 Q13255 2/20 0.31
GRM5 P41594 1/20 0.31
IRAK4 Q9NWZ3 7/20 0.31
KDM4E B2RXH2 1/20 0.31
BTK Q06187 1/20 0.30
CHRM4 P08173 1/20 0.30
GALR3 O60755 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19287695 0.80 KDM4E (0.36) ADORA3ADORA2AADORA1ADORA2BIRAK4
SCHEMBL7989472 0.79 KDM4E (0.33) TP53LMNAADORA3ADORA2AADORA1
SCHEMBL7989476 0.79 KDM4E (0.33) TP53LMNAADORA3ADORA2AADORA1
SCHEMBL23323316 0.77 TP53 (0.42) TP53LMNAGRM1GRM5
SCHEMBL7973702 0.77 TSHR (0.36) ADORA3ADORA2AADORA1ADORA2BBTK
SCHEMBL7970268 0.77 KDM4E (0.33) KDM4ECHRM4
SCHEMBL7971763 0.76 ADORA3 (0.39) ADORA3ADORA2AADORA1ADORA2BBTK
SCHEMBL7992282 0.75 KDM4E (0.34) IRAK4KDM4ECHRM4
SCHEMBL8490623 0.72 PRCP (0.46) ADORA3ADORA2AADORA1ADORA2BIRAK4
SCHEMBL8490628 0.72 PRCP (0.46) ADORA3ADORA2AADORA1ADORA2BIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6281221-B1 Substituted 1,3-dioxan-5-ylamino-hererocyclic compounds, processes for their preparation and their use as pest control compositions HOECHST SCERING AGREVO GMBH (DE) 2001-08-28 US disclosed
EP-0836603-A1 SUBSTITUTED 1,3-DIOXAN-5-YLAMINO HETEROCYCLIC COMPOUNDS, METHODS FOR PREPARING THEM AND THEIR USE AS PESTICIDES Hoechst Schering AgrEvo GmbH (DE) 1998-04-22 EP disclosed
WO-1997002264-A1 SUBSTITUTED 1,3-DIOXAN-5-YLAMINO HETEROCYCLIC COMPOUNDS, METHODS FOR PREPARING THEM AND THEIR USE AS PESTICIDES HOECHST SCHERING AGREVO GMBH (DE) 1997-01-23 WO disclosed