SCHEMBL7977997

SCHEMBL7977997

N#CN/C(=N\c1ccncc1)NCCOCCO

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LATS1 O95835 2/20 0.37
HRH4 Q9H3N8 4/20 0.35
CYP3A4 P08684 4/20 0.35
NAMPT P43490 4/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
CYP2D6 P10635 2/20 0.35
P2RX7 Q99572 2/20 0.34
CYP1A2 P05177 2/20 0.34
ABCC9 O60706 2/20 0.34
KCNJ11 Q14654 2/20 0.34
ALOX15 P16050 1/20 0.34
NFKB1 P19838 1/20 0.34
MAPK1 P28482 1/20 0.34
HIF1A Q16665 1/20 0.34
HSD17B10 Q99714 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
GLA P06280 1/20 0.34
BLM P54132 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7978001 1.00 LATS1 (0.37) LATS1HRH4CYP3A4NAMPTCYP2C9
SCHEMBL8195513 0.82 NAMPT (0.53) HRH4CYP3A4NAMPTCYP2C9CYP2C19
SCHEMBL8195515 0.82 NAMPT (0.53) HRH4CYP3A4NAMPTCYP2C9CYP2C19
SCHEMBL7098788 0.82 HRH4 (0.43) HRH4CYP3A4NAMPTCYP2C9CYP2C19
SCHEMBL8196333 0.81 ADRB2 (0.36) HRH4NAMPTLMNAIMPDH2
SCHEMBL8196331 0.81 ADRB2 (0.36) HRH4NAMPTLMNAIMPDH2
SCHEMBL8200604 0.81 NAMPT (0.35) HRH4NAMPTLMNAQPCTIMPDH2
SCHEMBL8195619 0.80 MEN1 (0.44) CYP3A4NAMPTCYP2C9CYP2C19CYP2D6
SCHEMBL8195623 0.80 MEN1 (0.44) CYP3A4NAMPTCYP2C9CYP2C19CYP2D6
SCHEMBL8919392 0.80 HRH4 (0.48) HRH4CYP3A4NAMPTCYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6255323-B1 Cyanoguanidine compounds SHIONOGI BIORESEARCH CORP. 2001-07-03 US disclosed
WO-2000061561-A1 CYANOGUANIDINE COMPOUNDS SHIONOGI BIORESEARCH CORP. (US) 2000-10-19 WO disclosed