SCHEMBL7978952

SCHEMBL7978952

CC(=O)N(c1cccc(F)c1)c1ccccn1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.45
HTT P42858 4/20 0.45
NPC1 O15118 3/20 0.45
RAB9A P51151 3/20 0.45
LMNA P02545 2/20 0.45
KDM4E B2RXH2 2/20 0.45
PTBP1 P26599 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
TP53 P04637 1/20 0.40
MAPK14 Q16539 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
PTGIR P43119 1/20 0.39
KMT2A Q03164 2/20 0.38
ACHE P22303 1/20 0.37
MEN1 O00255 1/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7969122 0.88 HTT (0.42) ALDH1A1HTTNPC1RAB9AKDM4E
SCHEMBL27511353 0.86 NPC1 (0.42) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL7985644 0.84 TRPM8 (0.42) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL7982503 0.84 S100A4 (0.48) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL7978872 0.83 HTT (0.40) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL19512684 0.83 NPSR1 (0.47) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL4613837 0.83 MAPT (0.44) HTTSMN1; SMN2NPSR1TP53KMT2A
SCHEMBL7978950 0.82 POLQ (0.47) ALDH1A1HTTLMNASMN1; SMN2CYP1A2
SCHEMBL30285727 0.82 NPC1 (0.40) ALDH1A1HTTNPC1RAB9ALMNA
SCHEMBL26186409 0.82 NPC1 (0.40) ALDH1A1HTTNPC1RAB9ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
CN-1252068-A 3-piperidyl-4-oxoquinazoline derivatives and pharmaceutical compositions containing the same JAPAN TOBACCO INC (JP) 2000-05-03 CN disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed