SCHEMBL7978872

SCHEMBL7978872

O=C(CF)N(c1cccc(F)c1)c1ccccn1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
PTGIR P43119 4/20 0.39
NPC1 O15118 2/20 0.39
LMNA P02545 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
PTGER4 P35408 1/20 0.37
PTGER3 P43115 1/20 0.37
PTGER2 P43116 1/20 0.37
PTGDR Q13258 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7982394 0.86 PTGIR (0.46) HTTPTGIRNPC1CYP1A2CYP2C9
SCHEMBL27511353 0.83 NPC1 (0.42) HTTPTGIRNPC1LMNACYP1A2
SCHEMBL7978952 0.83 ALDH1A1 (0.45) HTTPTGIRNPC1LMNACYP1A2
SCHEMBL7978997 0.76 HTT (0.41) HTTNPC1LMNARAB9AKMT2A
SCHEMBL7969122 0.71 HTT (0.42) HTTNPC1RAB9AKMT2ANPSR1
SCHEMBL7978994 0.71 NPSR1 (0.41) HTTPTGIRNPC1RAB9AKMT2A
SCHEMBL7980229 0.71 NPC1 (0.66) HTTPTGIRNPC1LMNACYP1A2
SCHEMBL7981944 0.71 PTGIR (0.46) HTTPTGIRNPC1RAB9AKMT2A
SCHEMBL7978941 0.69 TP53 (0.51) HTTPTGIRNPC1RAB9AKMT2A
SCHEMBL28682606 0.69 PTGIR (0.44) HTTPTGIRNPC1LMNARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6235730-B1 ANTICHOLESTEROL AGENT, ANTILIPEMIC AGENT JAPAN TOBACCO, INC. (JP) 2001-05-22 US disclosed
EP-0970954-A1 3-PIPERIDYL-4-OXOQUINAZOLINE DERIVATIVES AND MEDICINCAL COMPOSITIONS CONTAINING THE SAME JAPAN TOBACCO INC. (JP) 2000-01-12 EP disclosed