SCHEMBL7979370

SCHEMBL7979370

c1ccc(-c2cnc(Nc3cccc(-c4ncc[nH]4)c3)s2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 16/20 0.63
MTOR P42345 1/20 0.49
ADK P55263 1/20 0.49
NISCH Q9Y2I1 1/20 0.49
VCP P55072 1/20 0.48
ROCK1 Q13464 1/20 0.46
HDAC3 O15379 1/20 0.44
ABL1 P00519 1/20 0.44
PDGFRB P09619 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC7 Q8WUI4 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC10 Q969S8 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
HDAC9 Q9UKV0 1/20 0.44
HDAC5 Q9UQL6 1/20 0.44
CHEK1 O14757 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3651635 0.79 KDR (1.00) KDRROCK1
SCHEMBL7968277 0.78 ALOX5 (0.60) VCPHDAC6
SCHEMBL7967542 0.77 KDR (0.59) KDRROCK1ABL1PDGFRBCHEK1
SCHEMBL6335500 0.76 KDR (0.74) KDRROCK1
SCHEMBL6330184 0.74 KDR (1.00) KDRHDAC3ABL1PDGFRBHDAC4
SCHEMBL7981286 0.74 MTOR (0.48) KDRMTORADKNISCHVCP
SCHEMBL6330404 0.74 KDR (1.00) KDRROCK1
SCHEMBL7967444 0.73 MAPT (0.47) VCPHDAC6
SCHEMBL6332844 0.73 KDR (0.68) KDR
SCHEMBL6336629 0.73 KDR (0.69) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001087845-A2 N-CONTAINING HETEROCYCLIC COMPOUNDS AND THEIR USE AS 5-HT ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-11-22 WO disclosed