SCHEMBL7979453

SCHEMBL7979453

COc1ccccc1Oc1c(C(N)=O)nc(N2CCOCC2)nc1C(O)[C@H]1O[C@@H]2OC(C)(C)O[C@@H]2[C@H]2OC(C)(C)O[C@H]21

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.35
EDNRB P24530 9/20 0.34
EDNRA P25101 9/20 0.34
PIK3CB P42338 3/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 1/20 0.33
MTOR P42345 1/20 0.33
PIK3CG P48736 1/20 0.33
HTT P42858 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GPR55 Q9Y2T6 1/20 0.33
KDM4E B2RXH2 1/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R1 P27986 1/20 0.32
ATR Q13535 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7990192 0.81 PIK3CA (0.36) PIK3CAEDNRBEDNRAPIK3CBMAPT
SCHEMBL6586303 0.73 HTT (0.43) PIK3CAEDNRBEDNRAALDH1A1MAPT
SCHEMBL4068802 0.69 DHPS (0.50) EDNRBEDNRA
SCHEMBL7841637 0.67 EDNRB (0.54) EDNRBEDNRA
SCHEMBL5633057 0.65 MAPT (0.49) PIK3CAEDNRBEDNRAPIK3CBALDH1A1
SCHEMBL5653603 0.65 EDNRB (0.65) EDNRBEDNRA
SCHEMBL5631503 0.63 MAPT (0.49) PIK3CAPIK3CBALDH1A1MAPTMTOR
SCHEMBL5764886 0.63 EDNRB (0.53) EDNRBEDNRA
SCHEMBL6586305 0.61 DHPS (0.55) PIK3CAALDH1A1MAPTMTORLMNA
SCHEMBL4068803 0.61 DHPS (0.61) EDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001081338-A1 SUBSTITUTED SULFONYLAMINOPYRIMIDINES ACTELION PHARMACEUTICALS LTD (CH) 2001-11-01 WO disclosed