SCHEMBL7979742

SCHEMBL7979742

Nc1cccc2nc(CCO)cn12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
RAB9A P51151 5/20 0.34
MAPT P10636 5/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
NPC1 O15118 2/20 0.34
KMT2A Q03164 2/20 0.34
ADORA2A P29274 1/20 0.34
MEN1 O00255 1/20 0.34
KDM4E B2RXH2 3/20 0.33
GAA P10253 2/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
PDE10A Q9Y233 1/20 0.32
NUDT1 P36639 1/20 0.32
ALDH1A1 P00352 2/20 0.31
PTGS1 P23219 1/20 0.31
PTGS2 P35354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7980201 0.77 RAB9A (0.38) HTR2AHTR2CRAB9AMAPTSMN1; SMN2
SCHEMBL3021189 0.76 RAB9A (0.41) RAB9AMAPTSMN1; SMN2NPC1KMT2A
SCHEMBL7982683 0.71 GAA (0.47) MAPTKMT2AMEN1KDM4EGAA
SCHEMBL13218395 0.71 KDM4E (0.34) HTR2AHTR2CSMN1; SMN2NPC1KDM4E
SCHEMBL8373773 0.69 ALDH1A1 (0.40) RAB9ASMN1; SMN2NPC1KMT2AADORA2A
SCHEMBL7834962 0.69 PDE10A (0.59) RAB9AMAPTSMN1; SMN2NPC1KMT2A
SCHEMBL3734117 0.69 RAB9A (0.41) RAB9AMAPTSMN1; SMN2NPC1KMT2A
SCHEMBL7969411 0.69 KLKB1 (0.34) PDE10A
SCHEMBL5384818 0.69 PDE10A (0.47) RAB9AMAPTSMN1; SMN2NPC1KMT2A
SCHEMBL3035988 0.68 PTGS1 (0.51) HTR2AHTR2CMAPTKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174877-B1 EXCELLANT BACTERICIDES, ORAL ABSORBABILITY AND STABILITY; IMPROVE THE STABILITY TO RENAL DEHYDROPEPTIDASE I (DHP-I); 2-(2-(N-HETEROCYCLIC-ETHYLTHIO-) DERIVATIVES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-16 US disclosed
EP-0876370-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1998-11-11 EP disclosed
WO-1997025325-A1 CARBAPENEM COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-07-17 WO disclosed