SCHEMBL798024

SCHEMBL798024

O=C1NCCc2sc(Br)cc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 2/20 0.54
DBF4 Q9UBU7 1/20 0.54
PARP10 Q53GL7 12/20 0.46
PARP1 P09874 9/20 0.46
PARP11 Q9NR21 7/20 0.46
MAPK1 P28482 2/20 0.41
RAF1 P04049 1/20 0.41
MAP2K1 Q02750 1/20 0.41
PDPK1 O15530 1/20 0.39
F7 P08709 1/20 0.39
F3 P13726 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ACHE P22303 1/20 0.35
PRKD3 O94806 2/20 0.34
CDK1 P06493 2/20 0.34
CSNK1A1 P48729 2/20 0.34
CSNK1D P48730 2/20 0.34
CSNK1G2 P78368 2/20 0.34
CDK5 Q00535 2/20 0.34
PRKCQ Q04759 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18304962 0.89 CDC7 (0.44) CDC7DBF4PARP10PARP1PARP11
SCHEMBL23141727 0.81 CLK4 (0.39) CDC7DBF4PARP10PARP1PARP11
SCHEMBL12241446 0.78 CDC7 (0.54) CDC7DBF4PARP10PARP1PARP11
SCHEMBL25224674 0.76 PARP10 (0.40) CDC7DBF4PARP10PARP1PARP11
SCHEMBL25364126 0.74 CDC7 (0.50) CDC7DBF4PARP10PARP1PARP11
SCHEMBL12219888 0.74 CDC7 (0.50) CDC7DBF4PARP10PARP1PARP11
SCHEMBL23042702 0.72 PBRM1 (0.31) MAPK1RAF1MAP2K1
SCHEMBL18333426 0.71 CDC7 (0.76) CDC7DBF4PARP10PARP1PARP11
SCHEMBL390545 0.70 PARP10 (0.46) CDC7DBF4PARP10PARP1PARP11
SCHEMBL25204118 0.70 FABP6 (0.43) CDC7DBF4PARP10PARP1PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 31 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260070902-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2026-03-12 US disclosed
EP-4630402-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS F. Hoffmann-La Roche AG (CH) 2025-10-15 EP disclosed
CN-120091998-A Substituted bicyclic rings as HSET inhibitors 默克专利股份公司 2025-06-03 CN disclosed
US-20250144094-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF ERASCA, INC. 2025-05-08 US disclosed
EP-4433059-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF Erasca, Inc. (US) 2024-09-25 EP disclosed
WO-2024121013-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2024-06-13 WO disclosed
CN-113518779-B Thieno heterocyclic derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2024-03-15 CN disclosed
WO-2023215494-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF ERASCA, INC. (US) 2023-11-09 WO disclosed
CN-113493438-B Tetrahydroisoquinoline compounds 南京再明医药有限公司 2023-10-20 CN disclosed
EP-4216946-A1 PHARMACEUTICAL COMPOUNDS FOR THE TREATMENT OF COMPLEMENT MEDIATED DISORDERS Achillion Pharmaceuticals, Inc. (US) 2023-08-02 EP disclosed
WO-2016205534-A1 INHIBITORS OF PTP4A3 FOR THE TREATMENT OF CANCER LAZO JOHN S (US) 2016-12-22 WO disclosed
US-8946260-B2 17α-hydroxylase/C17,20-lyase inhibitors NOVARTIS AG (CH) 2015-02-03 US disclosed
US-8946260-B2 17α-hydroxylase/C17,20-lyase inhibitors NOVARTIS AG (CH) 2015-02-03 US disclosed
US-8946260-B2 17α-hydroxylase/C17,20-lyase inhibitors NOVARTIS AG (CH) 2015-02-03 US disclosed
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2014-02-13 US disclosed
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2014-02-13 US disclosed
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2014-02-13 US disclosed
EP-2627648-A1 17aHYDROXYLASE/C17,20-LYASE INHIBITORS Novartis AG (CH) 2013-08-21 EP disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed
WO-2012035078-A1 17α-HYDROXYLASE/C17,20-LYASE INHIBITORS NOVARTIS AG (CH) 2012-03-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250144094-A1 THIOPHENE ULK1/2 INHIBITORS AND THEIR USE THEREOF ULK1, ULK2, ULK3 CDC7 86/4885DBF4 1727/4885PARP10 547/4885
US-20260070902-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS CCR6, CCR1, CCR4 CDC7 1565/4885DBF4 3108/4885PARP10 3928/4885
US-20140045872-A1 17a-HYDROXYLASE/C17,20-LYASE INHIBITORS CYP17A1, CYP21A2, HSD17B1 CDC7 1205/4885DBF4 3433/4885PARP10 940/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.