SCHEMBL7980604

SCHEMBL7980604

O=C1CCCc2c(Cl)nsc21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 3/20 0.35
MAPK1 P28482 1/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
GAA P10253 1/20 0.34
PIK3CD O00329 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7977358 0.68 TSHR (0.32) SMN1; SMN2ALDH1A1
SCHEMBL7977027 0.66 RAB9A (0.35) SMN1; SMN2ALDH1A1MAPK1NPC1GAA
SCHEMBL29423714 0.60 ALDH1A1 (0.31) SMN1; SMN2ALDH1A1KDM4E
SCHEMBL167247 0.60 ALDH1A1 (0.61) SMN1; SMN2ALDH1A1MAPK1KDM4ENPC1
SCHEMBL6801673 0.58 DRD4 (0.45) SMN1; SMN2ALDH1A1KDM4EGAA
SCHEMBL16161354 0.57 HSD17B10 (0.37) SMN1; SMN2ALDH1A1MAPK1KDM4E
SCHEMBL14502277 0.57 ALDH1A1 (0.36) SMN1; SMN2ALDH1A1MAPK1KDM4E
SCHEMBL289021 0.57
SCHEMBL581560 0.57 MAPK1 (0.32) MAPK1KDM4E
SCHEMBL30375516 0.57 MAPK1 (0.32) MAPK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6174909-B1 FOR TREATING ANALGESIA, PSYCHOSIS, CONVULSIONS, EPILEPSY, ANXIETY, MUSCULAR AND MOVEMENT DISORDERS, SPASTIC DISORDERS OR SYMPTOMS OF HUNTINGTON'S OR PARKINSONS DISEASE H. LUNDBECK A/S (DK) 2001-01-16 US disclosed
US-5998613-A PSYCHOLOGICAL DISORDERS; ANALGESICS; ANTICONVULSANTS H. LUNDBECK A/S (DK) 1999-12-07 US disclosed
EP-0812318-A1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS H. LUNDBECK A/S (DK) 1997-12-17 EP disclosed
WO-1996026929-A1 4-AMINOTETRAHYDROBENZISOXAZOLE OR -ISOTHIAZOLE COMPOUNDS H. LUNDBECK A/S (DK) 1996-09-06 WO disclosed