SCHEMBL7980700

SCHEMBL7980700

Cc1c(C(=O)CCNc2ccccn2)sc2ccccc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.47
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
F10 P00742 1/20 0.43
NPC1 O15118 5/20 0.42
RAB9A P51151 5/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
RXFP1 Q9HBX9 2/20 0.42
PRNP P04156 1/20 0.42
CYP2C19 P33261 2/20 0.41
CYP1A2 P05177 2/20 0.39
ALDH1A1 P00352 2/20 0.39
LMNA P02545 1/20 0.39
MAPK10 P53779 1/20 0.39
TP53 P04637 1/20 0.39
ATM Q13315 1/20 0.39
LIMK1 P53667 1/20 0.39
NPSR1 Q6W5P4 3/20 0.38
KMT2A Q03164 2/20 0.38
CYP2D6 P10635 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7971233 0.82 MAPT (0.48) HSD11B1TAS1R3TAS1R1F10NPC1
Hydrochloric Acid SCHEMBL7987810 0.81 MAPT (0.47) HSD11B1TAS1R3TAS1R1F10NPC1
Hydrochloric Acid SCHEMBL7970754 0.78 HSD11B1 (0.45) HSD11B1F10NPC1RAB9ASMN1; SMN2
SCHEMBL7984156 0.76 HSD11B1 (0.61) HSD11B1SMN1; SMN2RXFP1PRNPCYP2C19
SCHEMBL7970877 0.72 HSD11B1 (0.51) HSD11B1F10NPC1RAB9ASMN1; SMN2
SCHEMBL13963145 0.72 HSD11B1 (0.62) HSD11B1F10SMN1; SMN2RXFP1PRNP
SCHEMBL13589546 0.72 CYP2C19 (0.56) NPC1RAB9ASMN1; SMN2CYP2C19CYP1A2
SCHEMBL4834908 0.72 HSD11B1 (0.62) HSD11B1F10SMN1; SMN2RXFP1PRNP
Hydrochloric Acid SCHEMBL7970822 0.71 HSD11B1 (0.46) HSD11B1NPC1RAB9ASMN1; SMN2RXFP1
SCHEMBL4775261 0.70 HSD11B1 (0.61) HSD11B1F10SMN1; SMN2RXFP1PRNP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2001007431-A2 BENZOTHIOPHENE DERIVATIVES ELI LILLY AND COMPANY (US) 2001-02-01 WO disclosed